Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50021279
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50206613(3-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-benzo...)
Affinity DataIC50: 350nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50206613(3-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-benzo...)
Affinity DataIC50: 400nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222818(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 600nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50206600(3-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-benzo...)
Affinity DataIC50: 700nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222823(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 800nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222820(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 900nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222815(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 900nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222823(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222824(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222824(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222817(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222818(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222827(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222823(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222824(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50095469([5-(1-Benzyl-1H-indazol-3-yl)-furan-2-yl]-methanol...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222821(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(4-...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50206600(3-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-benzo...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222818(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-isoni...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222825(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222825(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222826(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222822(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222825(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222822(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222827(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222815(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222827(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222820(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222820(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(3-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222815(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50095469([5-(1-Benzyl-1H-indazol-3-yl)-furan-2-yl]-methanol...)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222821(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(4-...)
Affinity DataIC50: 1.86E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222819(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222822(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222816(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222816(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222826(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50095469([5-(1-Benzyl-1H-indazol-3-yl)-furan-2-yl]-methanol...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222826(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222819(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human AGS cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222817(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Sk-Hep1 cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222821(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(4-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222819(2-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-fur...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222817(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-N-(2-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHypoxia-inducible factor 1-alpha(Human)
Molecular Cancer Research Center

Curated by ChEMBL
LigandPNGBDBM50222816(5-[2-(4-adamantan-1-yl-phenoxy)-acetylamino]-nicot...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of hypoxia induced HIF1-alpha transcriptional activity in human Hep3B cells by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed