Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50021270
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222728(cyclo(-L-Am7(S2Py)-A2in-L-Ala-D-Pro-) | CHEMBL3942...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222736(cyclo(-L-Am7(S2Py)-Aib-L-Ser(Bzl)-D-Pro-) | CHEMBL...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222732(cyclo(-L-Am7(S2Py)-Aib-L-Phe-D-Pro-) | (5S,11S,13a...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222728(cyclo(-L-Am7(S2Py)-A2in-L-Ala-D-Pro-) | CHEMBL3942...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222730(cyclo(-L-Am7(S2Py)-L-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222735(cyclo(-L-Am7(S2Py)-D-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222735(cyclo(-L-Am7(S2Py)-D-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222729(cyclo(-L-Am7(S2Py)-Aib-L-Ph5-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222738(cyclo(-L-Am7(S2Py)-Aib-L-Ph4-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222736(cyclo(-L-Am7(S2Py)-Aib-L-Ser(Bzl)-D-Pro-) | CHEMBL...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222730(cyclo(-L-Am7(S2Py)-L-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222732(cyclo(-L-Am7(S2Py)-Aib-L-Phe-D-Pro-) | (5S,11S,13a...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222733(cyclo(-L-Am7(S2Py)-Aib-L-Ser-D-Pro-) | CHEMBL39396...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222737(cyclo(-L-Am7(S2Py)-Aib-L-Ala-D-Tic-) | CHEMBL23858...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222737(cyclo(-L-Am7(S2Py)-Aib-L-Ala-D-Tic-) | CHEMBL23858...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222727((5S,11S,13aR)-5,8,8-trimethyl-11-[5-(pyridin-2-yld...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222729(cyclo(-L-Am7(S2Py)-Aib-L-Ph5-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222738(cyclo(-L-Am7(S2Py)-Aib-L-Ph4-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222733(cyclo(-L-Am7(S2Py)-Aib-L-Ser-D-Pro-) | CHEMBL39396...)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222728(cyclo(-L-Am7(S2Py)-A2in-L-Ala-D-Pro-) | CHEMBL3942...)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222727((5S,11S,13aR)-5,8,8-trimethyl-11-[5-(pyridin-2-yld...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222735(cyclo(-L-Am7(S2Py)-D-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222736(cyclo(-L-Am7(S2Py)-Aib-L-Ser(Bzl)-D-Pro-) | CHEMBL...)
Affinity DataIC50: 24nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222726(cyclo(-L-Am7(S2Py)-L-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222733(cyclo(-L-Am7(S2Py)-Aib-L-Ser-D-Pro-) | CHEMBL39396...)
Affinity DataIC50: 26nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222737(cyclo(-L-Am7(S2Py)-Aib-L-Ala-D-Tic-) | CHEMBL23858...)
Affinity DataIC50: 29nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222726(cyclo(-L-Am7(S2Py)-L-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 33nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222726(cyclo(-L-Am7(S2Py)-L-A1in-L-Ala-D-Pro-) | CHEMBL39...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222738(cyclo(-L-Am7(S2Py)-Aib-L-Ph4-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 36nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222732(cyclo(-L-Am7(S2Py)-Aib-L-Phe-D-Pro-) | (5S,11S,13a...)
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222729(cyclo(-L-Am7(S2Py)-Aib-L-Ph5-D-Pro-) | CHEMBL39138...)
Affinity DataIC50: 43nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222727((5S,11S,13aR)-5,8,8-trimethyl-11-[5-(pyridin-2-yld...)
Affinity DataIC50: 43nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222730(cyclo(-L-Am7(S2Py)-L-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 56nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222734(cyclo(-L-Am7(S2Py)-Aib-L-Phg-D-Pro-) | CHEMBL42873...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222731(cyclo(-L-Am7(S2Py)-D-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222731(cyclo(-L-Am7(S2Py)-D-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 71nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 6(Mouse)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222734(cyclo(-L-Am7(S2Py)-Aib-L-Phg-D-Pro-) | CHEMBL42873...)
Affinity DataIC50: 86nMAssay Description:Inhibition of mouse HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222734(cyclo(-L-Am7(S2Py)-Aib-L-Phg-D-Pro-) | CHEMBL42873...)
Affinity DataIC50: 88nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Graduate School of Life Science and Systems Engineering

Curated by ChEMBL
LigandPNGBDBM50222731(cyclo(-L-Am7(S2Py)-D-2MePhe-L-Ala-D-Pro-) | CHEMBL...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed