Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50021240
LigandPNGBDBM50222499(N-(3-chlorophenyl)-2-(pyridin-4-ylmethylamino)nico...)
Affinity DataKi:  2nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222500(N-(4-cyclohexylphenyl)-2-(pyridin-4-ylmethylamino)...)
Affinity DataKi:  2nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222501(N-(4-chloro-3-(trifluoromethyl)phenyl)-2-(pyridin-...)
Affinity DataKi:  4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222498(N-(3,5-bis(trifluoromethyl)phenyl)-2-(pyridin-4-yl...)
Affinity DataKi:  8nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222509(N-(4-chlorophenyl)-2-(pyridin-4-ylmethylamino)nico...)
Affinity DataKi:  8nMAssay Description:Inhibition of unphosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222512(2-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethyl)...)
Affinity DataKi:  9nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM15019(N-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]p...)
Affinity DataKi:  10nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50132151(N-(4-chlorophenyl)-2-(pyridin-4-ylmethylamino)benz...)
Affinity DataKi:  15nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222513(N-(3,4-dichlorophenyl)-2-(pyridin-4-ylmethylamino)...)
Affinity DataKi:  17nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222516(N-(4-butylphenyl)-2-(pyridin-4-ylmethylamino)nicot...)
Affinity DataKi:  19nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222503(N-biphenyl-4-yl-2-[(pyridin-4-ylmethyl)-amino]-nic...)
Affinity DataKi:  23nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222517(2-(pyridin-4-ylmethylamino)-N-(4-(trifluoromethoxy...)
Affinity DataKi:  23nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222504(ethyl 5-(3-(2-(pyridin-4-ylmethylamino)nicotinamid...)
Affinity DataKi:  29nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222508(2-(benzo[d][1,3]dioxol-5-ylmethylamino)-N-(4-pheno...)
Affinity DataKi:  38nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222496(2-(1H-indazol-6-ylamino)-N-(4-phenoxyphenyl)nicoti...)
Affinity DataKi:  70nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222507(N-biphenyl-3-yl-2-[(pyridin-4-ylmethyl)-amino]-nic...)
Affinity DataKi:  91nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222520(N-(3-ethylphenyl)-2-(pyridin-4-ylmethylamino)nicot...)
Affinity DataKi:  106nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222497(N-(4-chlorophenyl)-3-(pyridin-4-ylmethylamino)thio...)
Affinity DataKi:  120nMAssay Description:Inhibition of unphosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222522(2-(4-fluorophenylamino)-N-(4-phenoxyphenyl)nicotin...)
Affinity DataKi:  135nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222519(N-(4-chlorophenyl)-4-(pyridin-4-ylmethylamino)pyri...)
Affinity DataKi:  140nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222510(N-(3-phenoxyphenyl)-2-(pyridin-4-ylmethylamino)nic...)
Affinity DataKi:  259nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222515(2-(pyridin-4-ylmethylamino)-N-p-tolylnicotinamide ...)
Affinity DataKi:  320nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222523(5-bromo-N-(4-chlorophenyl)-2-(pyridin-4-ylmethylam...)
Affinity DataKi:  490nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222514(N-(3-(1-hydroxyethyl)phenyl)-2-(pyridin-4-ylmethyl...)
Affinity DataKi: >6.66E+3nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222506(N-(4-(4-methylpiperazin-1-yl)phenyl)-2-(pyridin-4-...)
Affinity DataKi: >6.66E+3nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222511(N-(4-chlorophenyl)-2-(pyridin-4-ylmethylamino)cycl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222505(N-(4-chlorophenyl)-3-(pyridin-4-ylmethylamino)pico...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222521(N-(4-chlorophenyl)-6-methyl-2-(pyridin-4-ylmethyla...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of unphosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222518(2-(benzo[b]thiophen-3-ylamino)-N-(4-phenoxyphenyl)...)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50222502(N-(2-phenoxyphenyl)-2-(pyridin-4-ylmethylamino)nic...)
Affinity DataKi: >2.00E+4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed