Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50021021
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220067(11H-2,5,11-triaza-benzo[a]trindene-1,3,4,6-tetraon...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220064(4,7,11-trihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220072(11-hydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220066(6,7-dihydro-1H-cyclopenta[a]pyrrolo[3,4-c]carbazol...)
Affinity DataIC50: 43nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50: 81nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220075(11-methylbenzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2...)
Affinity DataIC50: 107nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220065(4,7-dihydroxy-11-methylbenzo[a]pyrrolo[3,4-c]carba...)
Affinity DataIC50: 161nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220074(benzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2H,8H)-tet...)
Affinity DataIC50: 269nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220068(4,7-dihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2...)
Affinity DataIC50: 311nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50216165(1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,...)
Affinity DataIC50: 350nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50216157(11H-2,5,11,11b-Tetraaza-benzo[a]trindene-4,6-dione...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220063(4-hydroxy-11-methyl-7-hydroxysulfonyloxybenzo[a]py...)
Affinity DataIC50: 893nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220073(4-hydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H...)
Affinity DataIC50: 904nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220069(4-hydroxy-7-hydroxysulfonyloxybenzo[a]pyrrolo[3,4-...)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220070(7-tert-butylcarbonyloxy-4-hydroxybenzo[a]pyrrolo[3...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50220064(4,7,11-trihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed