Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50003863
LigandPNGBDBM50476682(CHEMBL428712 | PB-43)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476678(CHEMBL395222)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13328(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50: 3nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476685(CHEMBL232104)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM13324(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13327(N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476680(CHEMBL234757)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13335(N-tert-butyl-2-({6-cyano-1-[(1-methyl-1H-imidazol-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476679(CHEMBL232523)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476681(CHEMBL234151 | PB-91)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476676(CHEMBL231662)
Affinity DataIC50: 7nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476675(CHEMBL233742)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476677(CHEMBL394086 | PB-90)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13330(N-[(6-chloro-2,1,3-benzothiadiazol-5-yl)methyl]-N-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476674(CHEMBL394407 | PB-95)
Affinity DataIC50: 16nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476684(CHEMBL392237)
Affinity DataIC50: 25nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM50476683(CHEMBL234161)
Affinity DataIC50: 105nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13329(Pyridine-2-sulfonic Acid (1-Bromonaphthalen-2-ylme...)
Affinity DataIC50: 440nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
LigandPNGBDBM13326(N-[(1-bromonaphthalen-2-yl)methyl]-N-{6-cyano-1-[(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of protein farnesyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed