Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50021013
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(N-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219946(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenyl)pipe...)
Affinity DataIC50: 0.300nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219943(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219940(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219944(N-((1r,4r)-4-(2-(4-(4-bromo-2-methoxyphenyl)pipera...)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219947(N-((1r,4r)-4-(2-(4-(3-cyanophenyl)piperazin-1-yl)e...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219945(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219935(N-[4-(4-{2-[4-(3-cyano-5-trifluoromethyl-phenyl)-p...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219949(3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219942(N-((1r,4r)-4-(2-(4-(2,5-dichlorophenylamino)piperi...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219948(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219938(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenoxy)pip...)
Affinity DataIC50: 2.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219937(4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219936(4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50: 3.30nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219934(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 3.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(N-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219941(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219940(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 4.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219949(3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)pheno...)
Affinity DataIC50: 5.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219950(3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50: 5.80nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219942(N-((1r,4r)-4-(2-(4-(2,5-dichlorophenylamino)piperi...)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219937(4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219950(3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219943(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219936(4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluorome...)
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219944(N-((1r,4r)-4-(2-(4-(4-bromo-2-methoxyphenyl)pipera...)
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219946(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenyl)pipe...)
Affinity DataIC50: 29nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219945(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219935(N-[4-(4-{2-[4-(3-cyano-5-trifluoromethyl-phenyl)-p...)
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219941(N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phe...)
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219934(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219947(N-((1r,4r)-4-(2-(4-(3-cyanophenyl)piperazin-1-yl)e...)
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219938(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenoxy)pip...)
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219948(N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)benzyl)pipe...)
Affinity DataIC50: 91nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed