Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50025407
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
University of Bern

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataEC50:  191nMAssay Description:Activity at rat wild type GABAA alpha-1-beta-2-gamma-2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode volt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
University of Bern

Curated by ChEMBL
LigandPNGBDBM50242613(8-Isothiocyanato-5-methyl-6-oxo-5,6-dihydro-4H-2,5...)
Affinity DataEC50:  250nMAssay Description:Activity at rat wild type GABAA alpha-1-beta-2-gamma-2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode volt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
University of Bern

Curated by ChEMBL
LigandPNGBDBM26267(RO-154513 | Ro15-4513 | ethyl 12-azido-8-methyl-9-...)
Affinity DataEC50:  1.10nMAssay Description:Activity at rat wild type GABAA alpha-1-beta-2-gamma-2 receptor expressed in xenopus oocytes assessed as GABA-elicited response by two electrode volt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Human)
University of Bern

Curated by ChEMBL
LigandPNGBDBM50242613(8-Isothiocyanato-5-methyl-6-oxo-5,6-dihydro-4H-2,5...)
Affinity DataKd:  878nMAssay Description:Displacement of [3H]Ro15-1788 from rat GABAA alpha-1-beta-2-gamma-2 receptor expressed in HEK293 cells after 1 hr assessed as residual binding by liq...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed