Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 4673
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328726(CHEMBL1229814 | 4-Substituted Pyrrolidine Ring, 18...)
Affinity DataIC50: 0.160nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328728(CHEMBL1269832 | 4-Substituted Pyrrolidine Ring, 13...)
Affinity DataIC50: 0.380nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81692(4-Substituted Pyrrolidine Ring, 14)
Affinity DataIC50: 0.75nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81698(4-Substituted Pyrrolidine Ring, 35)
Affinity DataIC50: 1nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81693(4-Substituted Pyrrolidine Ring, 17 | 4-Substituted...)
Affinity DataIC50: 1.20nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328726(CHEMBL1229814 | 4-Substituted Pyrrolidine Ring, 18...)
Affinity DataIC50: 1.70nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81695(4-Substituted Pyrrolidine Ring, 20)
Affinity DataIC50: 2.90nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81697(4-Substituted Pyrrolidine Ring, 34)
Affinity DataIC50: 4.30nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81696(4-Substituted Pyrrolidine Ring, 21)
Affinity DataIC50: 5nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328728(CHEMBL1269832 | 4-Substituted Pyrrolidine Ring, 13...)
Affinity DataIC50: 6.10nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81693(4-Substituted Pyrrolidine Ring, 17 | 4-Substituted...)
Affinity DataIC50: 7nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81699(4-Substituted Pyrrolidine Ring, 36)
Affinity DataIC50: 7.60nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328725(CHEMBL1271371 | P1 Phenyl Ring, 23 | 4-Substituted...)
Affinity DataIC50: 18nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81681(P1 Phenyl Ring, 22)
Affinity DataIC50: 33nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM50328725(CHEMBL1271371 | P1 Phenyl Ring, 23 | 4-Substituted...)
Affinity DataIC50: 36nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81682(P1 Phenyl Ring, 24)
Affinity DataIC50: 389nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81683(P1 Phenyl Ring, 25)
Affinity DataIC50: 516nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81684(P1 Phenyl Ring, 26)
Affinity DataIC50: 873nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81685(P1 Phenyl Ring, 27)
Affinity DataIC50: 951nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81691(P1 Phenyl Ring, 33)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81690(P1 Phenyl Ring, 32)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81689(P1 Phenyl Ring, 31)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81688(P1 Phenyl Ring, 30)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81687(P1 Phenyl Ring, 29)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Pfizer

LigandPNGBDBM81686(P1 Phenyl Ring, 28)
Affinity DataIC50: 4.00E+3nMAssay Description:FXa inhibition were determined by using an inhibition assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2011
Entry Details Article
PubMed