Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50020562
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215069(1,2,3-tris-[3-(4-(N-ethyl)-quinoliniumylamino)-pro...)
Affinity DataIC50: 86nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215071(N-[3-(4-quinolinylamino)-propyl]-N-[5-(4-quinoliny...)
Affinity DataIC50: 93nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215070(1,2,3-tri[3-(4-quinolinylamino)-propoxy]-benzene |...)
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215076(N-[3-(4-quinolinylamino)-propyl]-N-[5-(4-quinoliny...)
Affinity DataIC50: 130nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215075(N-[3-(4-quinolinylamino)-propyl]-3,5-di-[3-(4-quin...)
Affinity DataIC50: 220nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215072(N-(4-quinolinyl)-3,4-di-[3-(4-quinolinylamino)-pro...)
Affinity DataIC50: 270nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215068(N-[3-(4-quinolinylamino)-proyl]-3,5-di[3-(4-quinol...)
Affinity DataIC50: 360nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215073(N-[3-(4-quinolinyl)-aminopropyl]-N-(8-aminooctyl)-...)
Affinity DataIC50: 490nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215074(N-(3-guanidinopropyl)-N-[4-(4'-aminomethylphenyl)]...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215079(4,4'bis(guanidinomethyl)-cis-stilbene | CHEMBL2291...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215078(N-(3-guanidinopropyl)-N(8-aminooctyl)-3-[(N'-(N''-...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSmall conductance calcium-activated potassium channel protein 3(Rat)
University College London

Curated by ChEMBL
LigandPNGBDBM50215077(N-(3-guanidinopropyl)-N-(8-aminooctyl)-3-[N'-(N''-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of SKca channel-mediated after-hypepolarization in rat sympathetic neuronsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed