Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50003872
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476855(CHEMBL232112)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476850(CHEMBL232114)
Affinity DataKi:  6.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476852(CHEMBL231917)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476848(CHEMBL231916)
Affinity DataKi:  9.20nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476853(CHEMBL398059)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476851(CHEMBL231918)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476854(CHEMBL232113)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476849(CHEMBL231915)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]IMPY from beta amyloid plaque in human brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed