Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003828
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476305(CHEMBL2068511)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476305(CHEMBL2068511)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476304(CHEMBL2068512)
Affinity DataIC50: 460nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476304(CHEMBL2068512)
Affinity DataIC50: 480nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050517(N-alkyl Gly-boro-Pro derivative | Boronic acid der...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050517(N-alkyl Gly-boro-Pro derivative | Boronic acid der...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50171653(N-alkyl Gly-boro-Pro derivative | CHEMBL196120)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human placental DPP4 at pH 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50171653(N-alkyl Gly-boro-Pro derivative | CHEMBL196120)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human placental DPP4 at pH 8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476305(CHEMBL2068511)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50476304(CHEMBL2068512)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human placental DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed