Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50003825
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476276(CHEMBL390561)
Affinity DataKi:  3.60nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476283(CHEMBL227921)
Affinity DataKi:  4.5nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476279(CHEMBL227817)
Affinity DataKi:  5nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476277(CHEMBL1162947)
Affinity DataKi:  6.80nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476284(CHEMBL227869)
Affinity DataKi:  6.80nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476280(CHEMBL224148)
Affinity DataKi:  7.5nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476282(CHEMBL227750)
Affinity DataKi:  7.5nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476278(CHEMBL224149)
Affinity DataKi:  8.5nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476274(CHEMBL224147)
Affinity DataKi:  9nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476275(CHEMBL226662)
Affinity DataKi:  14nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476281(CHEMBL227923)
Affinity DataKi:  16nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50476273(CHEMBL228094)
Affinity DataKi:  21nMAssay Description:Displacement of [15I]IMPY from Abeta peptide plaques in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed