Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50003824
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50209771(Dihydro-quinolinone | 3,4-dihydroquinolin-2(1H)-on...)
Affinity DataIC50: 0.740nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 2 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50045333(CHEBI:90705 | SB-203580)
Affinity DataIC50: 56nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476266(CHEMBL388106)
Affinity DataIC50: 500nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476263(CHEMBL388130)
Affinity DataIC50: 900nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476272(CHEMBL227884)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476269(CHEMBL226972)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476264(CHEMBL425494)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476270(CHEMBL389508)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476271(CHEMBL228075)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476267(CHEMBL227692)
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476268(CHEMBL227609)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 11/12/13/14(Human)
Eberhard-Karls-University T£Bingen

Curated by ChEMBL
LigandPNGBDBM50476265(CHEMBL375948)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mitogen-activated protein kinase p38 at 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed