Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50025156
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260268(rPKPfQwFwLL-NH2 | CHEMBL501261)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260271(RwFwLL-NH2 | CHEMBL500703)
Affinity DataIC50: 12nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260270(KwFwLL-NH2 | CHEMBL506986)
Affinity DataIC50: 13nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260275(AwFwLL-NH2 | CHEMBL509976)
Affinity DataIC50: 15nMAssay Description:Agonist activity at human wild type ghrelin receptor expressed in african green monkey COS7 cells assessed as stimulation of constitutively stimulate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260275(AwFwLL-NH2 | CHEMBL509976)
Affinity DataIC50: 15nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260268(rPKPfQwFwLL-NH2 | CHEMBL501261)
Affinity DataIC50: 18nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260271(RwFwLL-NH2 | CHEMBL500703)
Affinity DataIC50: 21nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260270(KwFwLL-NH2 | CHEMBL506986)
Affinity DataIC50: 32nMAssay Description:Inverse agonist activity at human wild type ghrelin receptor expressed in african green monkey COS7 cells assessed as inhibition of constitutively st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260270(KwFwLL-NH2 | CHEMBL506986)
Affinity DataIC50: 36nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260275(AwFwLL-NH2 | CHEMBL509976)
Affinity DataIC50: 53nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260272(HwFwLL-NH2 | CHEMBL502208)
Affinity DataIC50: 58nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260274(DwFwLL-NH2 | CHEMBL449590)
Affinity DataIC50: 60nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260272(HwFwLL-NH2 | CHEMBL502208)
Affinity DataIC50: 68nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260273(DprwFwLL-NH2 | CHEMBL507636)
Affinity DataIC50: 112nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260276(QwFwLL-NH2 | CHEMBL499371)
Affinity DataIC50: 120nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260278(wFwGG-NH2 | CHEMBL444131)
Affinity DataIC50: 159nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260273(DprwFwLL-NH2 | CHEMBL507636)
Affinity DataIC50: 210nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260274(DwFwLL-NH2 | CHEMBL449590)
Affinity DataIC50: 260nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260269(wFwLL-NH2 | CHEMBL450217)
Affinity DataIC50: 530nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260278(wFwGG-NH2 | CHEMBL444131)
Affinity DataIC50: 540nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260276(QwFwLL-NH2 | CHEMBL499371)
Affinity DataIC50: 990nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260277(wFwAA-NH2 | CHEMBL447444)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [35S]MK677 from human ghrelin receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260277(wFwAA-NH2 | CHEMBL447444)
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50260269(wFwLL-NH2 | CHEMBL450217)
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist activity at human ghrelin receptor expressed in african green monkey COS7 cells assessed as constitutively stimulated inositol phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed