Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50003937
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50183273((S)-6-(3-chloro-2-fluorobenzyl)-1-(1-hydroxy-3-met...)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM107681(CHEMBL320261 | CHEMBL19977 | (2Z)-4-[3,5-bis(benzy...)
Affinity DataIC50: 200nMAssay Description:Inhibition of HIV1 integrase-mediated 3'-end processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477786(CHEMBL252700)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477782(CHEMBL252905)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477783(CHEMBL401579)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477784(CHEMBL254727)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477787(CHEMBL404423)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM107681(CHEMBL320261 | CHEMBL19977 | (2Z)-4-[3,5-bis(benzy...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50142737((E)-6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-hex-5-en...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV1 integrase-mediated 3'-end processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50142737((E)-6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-hex-5-en...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50420376(CHEMBL267855)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50477785(CHEMBL254527)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
K.L.E.S. College of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50123468([3-Benzyl-5-(1,1-dioxo-1lambda 6 -isothiazolidin-2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed