Compile Data Set for Download or QSAR
Report error Found 109 Enz. Inhib. hit(s) with all data for entry = 50019811
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50411311(CHEMBL2113267)
Affinity DataIC50: 560nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50411311(CHEMBL2113267)
Affinity DataIC50: 650nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50292287(CHEMBL465161 | ginkgolide-A | GINKGOLIDE A)
Affinity DataIC50: 690nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50411311(CHEMBL2113267)
Affinity DataIC50: 780nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50411311(CHEMBL2113267)
Affinity DataIC50: 1.30E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 1.70E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataIC50: 1.70E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50292287(CHEMBL465161 | ginkgolide-A | GINKGOLIDE A)
Affinity DataIC50: 1.90E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50292287(CHEMBL465161 | ginkgolide-A | GINKGOLIDE A)
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 2.40E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 2.40E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 30 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataIC50: 2.90E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208076(3,14-didehydroginkgolide A | CHEMBL373969)
Affinity DataIC50: 3.10E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208068((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 3.20E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208081((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 3.20E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataIC50: 3.70E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50292287(CHEMBL465161 | ginkgolide-A | GINKGOLIDE A)
Affinity DataIC50: 3.80E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208074(ginkgolide J | CHEMBL374004)
Affinity DataIC50: 4.20E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208068((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 4.60E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 4.70E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208060(10-methoxy-ginkgolide C | CHEMBL221823)
Affinity DataIC50: 5.20E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 5.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 3000 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208076(3,14-didehydroginkgolide A | CHEMBL373969)
Affinity DataIC50: 6.20E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208074(ginkgolide J | CHEMBL374004)
Affinity DataIC50: 6.40E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208074(ginkgolide J | CHEMBL374004)
Affinity DataIC50: 7.10E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208068((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 7.30E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208082((1R,3R,6R,7S,8S,9S,10S,11R,12R,13S,16S,17R)-9-azid...)
Affinity DataIC50: 7.40E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208081((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 7.60E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208060(10-methoxy-ginkgolide C | CHEMBL221823)
Affinity DataIC50: 7.80E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 8.20E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208085((3S,8R,12R,16S,17R,21S)-3-tert-butyl-17-hydroxy-16...)
Affinity DataIC50: 8.90E+3nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208076(3,14-didehydroginkgolide A | CHEMBL373969)
Affinity DataIC50: 9.50E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208060(10-methoxy-ginkgolide C | CHEMBL221823)
Affinity DataIC50: 9.80E+3nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208074(ginkgolide J | CHEMBL374004)
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208085((3S,8R,12R,16S,17R,21S)-3-tert-butyl-17-hydroxy-16...)
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208085((3S,8R,12R,16S,17R,21S)-3-tert-butyl-17-hydroxy-16...)
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208081((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 1.30E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208082((1R,3R,6R,7S,8S,9S,10S,11R,12R,13S,16S,17R)-9-azid...)
Affinity DataIC50: 1.70E+4nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208082((1R,3R,6R,7S,8S,9S,10S,11R,12R,13S,16S,17R)-9-azid...)
Affinity DataIC50: 2.90E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208059(CHEMBL412384)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208061((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-9-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208062((1R,6R,8S,11S)-8-tert-butyl-6,13-dimethoxy-2,4,14,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208059(CHEMBL412384)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208063(10-methoxymethyloxy-ginkgolide A | CHEMBL225470)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208062((1R,6R,8S,11S)-8-tert-butyl-6,13-dimethoxy-2,4,14,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208065(methyl 2-[(1R,6R,8S,11S,14E)-8-tert-butyl-6-hydrox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208066((1R,2R,3S,6S,8S,10R,11R)-10-tert-butyl-2,11,16-tri...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1-beta-GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208067(methyl (2R)-2-[(1S,2R,3S,6S,8S,10S)-10-tert-butyl-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208066((1R,2R,3S,6S,8S,10R,11R)-10-tert-butyl-2,11,16-tri...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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