Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019778
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50207586(2,6-bis(3-bromo-4-hydroxybenzylidene)cyclohexanone...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50207589(1,7-bis(3-carboxy-4-hydroxyphenyl)-1,6-heptadiene-...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50207587(1,7-bis(3-bis(3-bromo-4-hydroxyphenyl)-1,6-heptadi...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50067030(1,7-bis(3,4-dihydroxyphenyl)-5-hydroxyhepta-1,4,6-...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50067033(2,6-Bis-[1-(4-hydroxy-3-methoxy-phenyl)-meth-(E)-y...)
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50207588(2,6-bis(3-carboxy-4-hydroxybenzylidene)cyclohexano...)
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50067027(2,6-bis(3,4-dihydroxybenzylidene)cyclohexanone | 2...)
Affinity DataIC50: 2.33E+5nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50067040(CHEMBL116438 | 1,7-bis(4-hydroxy-3-methoxyphenyl)1...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of GST-p300 HAT assessed as histone acetylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed