Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50037934
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206074((+/-)-N-{2-[2-(1-methyl-pyrrolidin-2-yl)-ethylamin...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206073(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-6-yl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206064(N-[2-(1-benzyl-piperidin-4-ylamino)-benzothiazol-6...)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206065(N-{2-[1-(3-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206080(N-{2-[1-(4-fluoro-benzyl)-piperidin-4-ylamino]-ben...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206076(N-{2-[1-(4-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206082(N-(2-amino-benzothiazol-6-yl)-thiophene-2-carboxam...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206070(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-6-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206067(N-(2-amino-benzothiazol-5-yl)-thiophene-2-carboxam...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206066(N-(2-{1-[2-(3H-imidazol-4-yl)-ethyl]-piperidin-4-y...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206075(4-(4-{6-[(thiophene-2-carboximidoyl)-amino]-benzot...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206079(N-[2-(1-benzyl-piperidin-4-ylamino)-benzothiazol-5...)
Affinity DataIC50: 400nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206064(N-[2-(1-benzyl-piperidin-4-ylamino)-benzothiazol-6...)
Affinity DataIC50: 500nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206066(N-(2-{1-[2-(3H-imidazol-4-yl)-ethyl]-piperidin-4-y...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206071(N-{2-[1-(4-fluoro-benzyl)-piperidin-4-ylamino]-ben...)
Affinity DataIC50: 800nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206070(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-6-...)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206073(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-6-yl...)
Affinity DataIC50: 900nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206072(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-5-yl...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206081(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-5-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206065(N-{2-[1-(3-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206073(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-6-yl...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206077(1-(2-amino-benzothiazol-6-yl)-2-ethyl-isothiourea ...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206070(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-6-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206074((+/-)-N-{2-[2-(1-methyl-pyrrolidin-2-yl)-ethylamin...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206069(N-{2-[1-(tetrahydro-pyran-4-yl)-piperidin-4-ylamin...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206068(N-(2-{1-[2-(4-Bromo-phenyl)-ethyl]-piperidin-4-yla...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206067(N-(2-amino-benzothiazol-5-yl)-thiophene-2-carboxam...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206082(N-(2-amino-benzothiazol-6-yl)-thiophene-2-carboxam...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206073(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-6-yl...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206065(N-{2-[1-(3-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206068(N-(2-{1-[2-(4-Bromo-phenyl)-ethyl]-piperidin-4-yla...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206066(N-(2-{1-[2-(3H-imidazol-4-yl)-ethyl]-piperidin-4-y...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206078(1-(2-amino-benzothiazol-5-yl)-2-ethyl-isothiourea ...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206068(N-(2-{1-[2-(4-Bromo-phenyl)-ethyl]-piperidin-4-yla...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206066(N-(2-{1-[2-(3H-imidazol-4-yl)-ethyl]-piperidin-4-y...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206063(4-(4-{6-[(thiophene-2-carboximidoyl)-amino]-benzot...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206075(4-(4-{6-[(thiophene-2-carboximidoyl)-amino]-benzot...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206068(N-(2-{1-[2-(4-Bromo-phenyl)-ethyl]-piperidin-4-yla...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206076(N-{2-[1-(4-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206072(N-[2-(2-pyridin-2-yl-ethylamino)-benzothiazol-5-yl...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206066(N-(2-{1-[2-(3H-imidazol-4-yl)-ethyl]-piperidin-4-y...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human inducible NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206064(N-[2-(1-benzyl-piperidin-4-ylamino)-benzothiazol-6...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, brain(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206065(N-{2-[1-(3-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of rat neuronal NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206080(N-{2-[1-(4-fluoro-benzyl)-piperidin-4-ylamino]-ben...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, inducible(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206076(N-{2-[1-(4-methoxy-benzyl)-piperidin-4-ylamino]-be...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human inducible NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206070(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-6-...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206077(1-(2-amino-benzothiazol-6-yl)-2-ethyl-isothiourea ...)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206081(N-[2-(2-morpholin-4-yl-ethylamino)-benzothiazol-5-...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Human)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206078(1-(2-amino-benzothiazol-5-yl)-2-ethyl-isothiourea ...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetNitric oxide synthase, endothelial(Rat)
Neuraxon

Curated by ChEMBL
LigandPNGBDBM50206064(N-[2-(1-benzyl-piperidin-4-ylamino)-benzothiazol-6...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of rat endothelial NOS activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 77 total ) | Next | Last >>
Jump to: