Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50019483
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205216((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205202(3-((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205133((S)-1-((3S,5S)-3-propylpyrrolidine-5-carbonyl)pyrr...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205219((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205128((S)-1-((3S,5S)-3-allylpyrrolidine-5-carbonyl)pyrro...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205214((2S)-1-{[(2S,4R)-4-(2-hydroxyethyl)-2-pyrrolidinyl...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205200((2S)-1-{[(2S,4S)-4-(1-azetidinylcarbonyl)-2-pyrrol...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205209((2S)-1-{[(2S,4S)-4-(4-morpholinylcarbonyl)-2-pyrro...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205215((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205224(2-((3R,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205223((2S)-1-{[(2S,4S)-4-(4-thiomorpholinylcarbonyl)-2-p...)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205210((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205212((2S)-1-{[(2S,4S)-4-(1-piperidinylcarbonyl)-2-pyrro...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205208((2S)-1-{[(2S,4S)-4-(1-pyrrolidinylcarbonyl)-2-pyrr...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205213(2S)-1-{[(2S,4S,5S)-4-(1,3-dihydro-2H-isoindol-2-yl...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205221((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205218((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205222((2S)-1-{[(2S,4S,5S)-5-methyl-4-(4-thiomorpholinylc...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205217((2S)-1-{[(2S,4S)-4-(hydroxymethyl)-2-pyrrolidinyl]...)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205211((2S)-1-{[(2S,4S,5S)-5-Methyl-4-(1-pyrrolidinylcarb...)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205204((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205203((2S)-1-{[(2S,4S)-4-(1-azepanylcarbonyl)-2-pyrrolid...)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205206((2S,3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205220((2S)-1-{[(2S,4S)-4-(1-azocanylcarbonyl)-2-pyrrolid...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205226((2S)-1-{[(2S,4S,5S)-5-methyl-4-(1-piperidinylcarbo...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205207((2S)-1-{[(2S,4S,5S)-4-(1-azetidinylcarbonyl)-5-met...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205205((2S,3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205225(((3R,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM11056(CHEMBL381626 | (2S)-1-[(2S)-pyrrolidin-2-ylcarbony...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205201((2S)-1-{[(2S,4S,5S)-5-methyl-4-(4-morpholinylcarbo...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed