Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50019351
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203825(Tyr-Pro-Phe-D-2-Nal-NH2 | CHEMBL375070)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203829(Dmt-Pro-Trp-D-1-Nal-NH2 | CHEMBL375068)
Affinity DataEC50:  1.20nMAssay Description:Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataEC50:  0.0400nMAssay Description:Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataEC50:  0.00100nMAssay Description:Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203822(Tyr-Pro-Trp-D-1-Nal-NH2 | CHEMBL219108)
Affinity DataEC50:  82nMAssay Description:Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203826(Tyr-Pro-Trp-D-2-Nal-NH2 | CHEMBL267211)
Affinity DataEC50:  248nMAssay Description:Activity at mu opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203827(Dmt-Pro-Phe-D-1-Nal-NH2 | CHEMBL385583)
Affinity DataEC50:  3.60nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203826(Tyr-Pro-Trp-D-2-Nal-NH2 | CHEMBL267211)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203822(Tyr-Pro-Trp-D-1-Nal-NH2 | CHEMBL219108)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203823(Dmt-Pro-Trp-D-2-Nal-NH2 | CHEMBL218433)
Affinity DataEC50:  29nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50232769(Dmt-Pro-Phe-D-2-Nal-NH2 | CHEMBL254919)
Affinity DataEC50:  16nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataEC50: <0.0100nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203828(Tyr-Pro-Phe-D-1-Nal-NH2 | CHEMBL375069)
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Medical University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataEC50:  932nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Medical University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 7.70nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Medical University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 15nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203829(Dmt-Pro-Trp-D-1-Nal-NH2 | CHEMBL375068)
Affinity DataIC50: 16nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Medical University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 17nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Medical University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 26nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203826(Tyr-Pro-Trp-D-2-Nal-NH2 | CHEMBL267211)
Affinity DataIC50: 3.47E+3nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203822(Tyr-Pro-Trp-D-1-Nal-NH2 | CHEMBL219108)
Affinity DataIC50: 4.18E+3nMAssay Description:Agonist activity at mu opioid receptor by inhibition of electrically evoked muscle contraction in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203828(Tyr-Pro-Phe-D-1-Nal-NH2 | CHEMBL375069)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203827(Dmt-Pro-Phe-D-1-Nal-NH2 | CHEMBL385583)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50232769(Dmt-Pro-Phe-D-2-Nal-NH2 | CHEMBL254919)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203823(Dmt-Pro-Trp-D-2-Nal-NH2 | CHEMBL218433)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50232769(Dmt-Pro-Phe-D-2-Nal-NH2 | CHEMBL254919)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203823(Dmt-Pro-Trp-D-2-Nal-NH2 | CHEMBL218433)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Medical University

Curated by ChEMBL
LigandPNGBDBM50203827(Dmt-Pro-Phe-D-1-Nal-NH2 | CHEMBL385583)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed