Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50019126
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202047(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-isopropylph...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202056(cis-3-{4-[1-(4-tert-butylcyclohexyl)-3-(4-trifluor...)
Affinity DataIC50: 47nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50144009(3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluorome...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202051(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(2-cyano...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50144009(3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluorome...)
Affinity DataIC50: 56nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202041(trans-3-{4-[3-(3,5-bistrifluoromethylphenyl)-1-(4-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202029(3-(4-((1-(4-isopropylcyclohexyl)-3-(4-(trifluorome...)
Affinity DataIC50: 59nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202039(3-(4-((1-(4-cyclohexylphenyl)-3-(4-(trifluorometho...)
Affinity DataIC50: 61nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202050(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(3,5-dic...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202060(3-{4-[1-(4-tert-butylphenyl)-3-(4-trifluoromethoxy...)
Affinity DataIC50: 96nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202038(3-(4-{[N-(5-chlorobenzo[b]thiophen-3-carbonyl)-N-(...)
Affinity DataIC50: 116nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50: 122nMAssay Description:Inhibition of rat glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202042(3-{4-[1-(4-propylcyclohexyl)-3-(4-trifluoromethoxy...)
Affinity DataIC50: 122nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202030(3-(4-((1-(4,4-dipropylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 137nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202045(trans-3-{4-[1-(4-tert-butylcyclohexyl)-3-(4-cyclop...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202035(3-(4-((1-(heptan-3-yl)-3-(4-(trifluoromethoxy)phen...)
Affinity DataIC50: 141nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202026(trans-3-{4-[3-(2-bromo-4-trifluoromethoxyphenyl)-1...)
Affinity DataIC50: 153nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202023(3-(4-((1-(4-cyclohexylphenyl)-3-(3-nitrophenyl)ure...)
Affinity DataIC50: 167nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202034(3-(4-((3-(4-butylphenyl)-1-(2,3-dihydro-1H-inden-2...)
Affinity DataIC50: 179nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202037(trans 3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(cycl...)
Affinity DataIC50: 182nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202024(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-cyano...)
Affinity DataIC50: 215nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202025(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(3,4-dic...)
Affinity DataIC50: 226nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202044(3-(4-((1-(2,3-dihydro-1H-inden-2-yl)-3-(4-(trifluo...)
Affinity DataIC50: 262nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202057(3-(4-((1-(4-phenoxycyclohexyl)-3-(4-(trifluorometh...)
Affinity DataIC50: 528nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202043(3-(4-((1-(4-cyclopropylidenecyclohexyl)-3-(4-(trif...)
Affinity DataIC50: 571nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202049(3-(4-((1-(4-(diethylcarbamoyl)cyclohexyl)-3-(4-(tr...)
Affinity DataIC50: 782nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202046(1-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50144009(3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(4-trifluorome...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GLP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202032(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-cyano...)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202033(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-phenylur...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202040(3-{4-[1-(1,4-dioxa-spiro[4.5]dec-8-yl)-3-(4-triflu...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202062(2-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50411232(CHEMBL2113259)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202036(trans-3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(diet...)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202059(1-(4-((2-(hydroxyamino)-2-oxoethyl)carbamoyl)benzy...)
Affinity DataIC50: 2.96E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of GLP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202022(3-(4-((2-chloro-N-(3,3-diphenylpropyl)nicotinamido...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202052(3-(4-((1-(4-(methylcarbamoyl)cyclohexyl)-3-(4-(tri...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202048(4-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202055(3-(4-((1-(4-((cyclopropylmethyl)carbamoyl)cyclohex...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202054(1-(4-((3-methoxypropyl)carbamoyl)benzyl)-1-(4-tert...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202053(3-(4-((1-(4-methoxycyclohexyl)-3-(4-(trifluorometh...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202028(4-(1-(4-((2-carboxyethyl)carbamoyl)benzyl)-3-(4-(t...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202027(1-(4-((3-amino-3-oxopropyl)carbamoyl)benzyl)-1-(4-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202061(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human cloned glucagon receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50202022(3-(4-((2-chloro-N-(3,3-diphenylpropyl)nicotinamido...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GLP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed