Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50019055
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201160(7-(4-hydroxyphenyl)benzo[b]thiophene-4-carbaldehyd...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201159(4-(3-fluoro-4-hydroxyphenyl)-1-naphthaldehyde oxim...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201158(4-(4-hydroxyphenyl)benzo[b]thiophene-7-carbaldehyd...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201164(4-(4-HYDROXYPHENYL)-1-NAPHTHALDEHYDE OXIME | CHEMB...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201161(1-(3-fluoro-4-hydroxyphenyl)-2-methyl-1H-indole-3-...)
Affinity DataIC50: 8.05nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201156(3,5-dichloro-3'-fluoro-4'-hydroxy-biphenyl-4-carba...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201163(4-(4-hydroxyphenyl)benzofuran-7-carbaldehyde oxime...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201155(1-(4-hydroxyphenyl)-2-methyl-1H-indole-3-carbaldeh...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201158(4-(4-hydroxyphenyl)benzo[b]thiophene-7-carbaldehyd...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201160(7-(4-hydroxyphenyl)benzo[b]thiophene-4-carbaldehyd...)
Affinity DataIC50: 37nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201164(4-(4-HYDROXYPHENYL)-1-NAPHTHALDEHYDE OXIME | CHEMB...)
Affinity DataIC50: 95nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201159(4-(3-fluoro-4-hydroxyphenyl)-1-naphthaldehyde oxim...)
Affinity DataIC50: 148nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201163(4-(4-hydroxyphenyl)benzofuran-7-carbaldehyde oxime...)
Affinity DataIC50: 155nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201162(1-(4-hydroxyphenyl)-1H-indole-3-carbaldehyde oxime...)
Affinity DataIC50: 202nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201155(1-(4-hydroxyphenyl)-2-methyl-1H-indole-3-carbaldeh...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201156(3,5-dichloro-3'-fluoro-4'-hydroxy-biphenyl-4-carba...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201161(1-(3-fluoro-4-hydroxyphenyl)-2-methyl-1H-indole-3-...)
Affinity DataIC50: 298nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 395nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201157(7-(4-hydroxyphenyl)benzofuran-4-carbaldehyde oxime...)
Affinity DataIC50: 457nMAssay Description:Inhibition of human ERbeta by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201157(7-(4-hydroxyphenyl)benzofuran-4-carbaldehyde oxime...)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201162(1-(4-hydroxyphenyl)-1H-indole-3-carbaldehyde oxime...)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of human ERalpha by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed