Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 2327
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.20nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.40nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 25nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19463(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-propyl-3,4-dih...)
Affinity DataIC50: 29nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19469(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(2-methylpropy...)
Affinity DataIC50: 37nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19460(CHEMBL376915 | YS04 | (2S)-5,7-dihydroxy-2-(4-hydr...)
Affinity DataIC50: 57nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19468(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methylbutyl...)
Affinity DataIC50: 59nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19460(CHEMBL376915 | YS04 | (2S)-5,7-dihydroxy-2-(4-hydr...)
Affinity DataIC50: 68nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19465(8-heptyl-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dih...)
Affinity DataIC50: 69nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19469(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(2-methylpropy...)
Affinity DataIC50: 80nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19464(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-pentyl-3,4-dih...)
Affinity DataIC50: 97nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19466(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-nonyl-3,4-dihy...)
Affinity DataIC50: 113nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19468(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methylbutyl...)
Affinity DataIC50: 140nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19470(8-(2,2-dimethylpropyl)-5,7-dihydroxy-2-(4-hydroxyp...)
Affinity DataIC50: 141nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19463(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-propyl-3,4-dih...)
Affinity DataIC50: 155nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19470(8-(2,2-dimethylpropyl)-5,7-dihydroxy-2-(4-hydroxyp...)
Affinity DataIC50: 216nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19471(8-benzyl-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dih...)
Affinity DataIC50: 244nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19464(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-pentyl-3,4-dih...)
Affinity DataIC50: 383nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19465(8-heptyl-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dih...)
Affinity DataIC50: 392nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19467(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-undecyl-3,4-di...)
Affinity DataIC50: 421nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19466(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-nonyl-3,4-dihy...)
Affinity DataIC50: 436nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19471(8-benzyl-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dih...)
Affinity DataIC50: 503nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19462(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-methyl-3,4-dih...)
Affinity DataIC50: 863nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19467(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-undecyl-3,4-di...)
Affinity DataIC50: 1.02E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 1.15E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19462(5,7-dihydroxy-2-(4-hydroxyphenyl)-8-methyl-3,4-dih...)
Affinity DataIC50: 5.25E+3nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
Ghent University

LigandPNGBDBM19461(5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro-2H-1...)
Affinity DataIC50: 1.35E+4nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Ghent University

LigandPNGBDBM19461(5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro-2H-1...)
Affinity DataIC50: 7.23E+4nMpH: 7.6 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated polyvinyltoluene scintillation beads (Amersham) and biot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2007
Entry Details Article
PubMed