Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50037928
TargetMatrix metalloproteinase-9(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM18050(MTX | cid_126941 | Methotrexate | 2-[(4-{[(2,4-dia...)
Affinity DataIC50: 9nMAssay Description:Inhibition of DHFR using dihydrofolic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM18050(MTX | cid_126941 | Methotrexate | 2-[(4-{[(2,4-dia...)
Affinity DataIC50: 35nMAssay Description:Inhibition of DHFR using folic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199731(methotrexate gamma-hydroxamic acid | CHEMBL244883)
Affinity DataIC50: 70nMAssay Description:Inhibition of DHFR using dihydrofolic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrilysin(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM8465(CGS 27023 | CHEMBL514138 | hydroxamate analogue 1 ...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199735(methotrexate gamma-L-proline-hydroxamic acid | CHE...)
Affinity DataIC50: 120nMAssay Description:Inhibition of DHFR using dihydrofolic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199735(methotrexate gamma-L-proline-hydroxamic acid | CHE...)
Affinity DataIC50: 130nMAssay Description:Inhibition of DHFR using folic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 170nMAssay Description:Inhibition of DHFR using dihydrofolic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199731(methotrexate gamma-hydroxamic acid | CHEMBL244883)
Affinity DataIC50: 170nMAssay Description:Inhibition of DHFR using folic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetDihydrofolate reductase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 250nMAssay Description:Inhibition of DHFR using folic acid substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrilysin(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199734(folate gamma-L-phenylalaninehydroxamic acid | CHEM...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199734(folate gamma-L-phenylalaninehydroxamic acid | CHEM...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of human recombinant MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrilysin(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199734(folate gamma-L-phenylalaninehydroxamic acid | CHEM...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of human recombinant MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199733(methotrexate gamma-L-phenylalaninehydroxamic acid ...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human recombinant MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199734(folate gamma-L-phenylalaninehydroxamic acid | CHEM...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human recombinant MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetMatrilysin(Human)
Instituto Superior T£Cnico

Curated by ChEMBL
LigandPNGBDBM50199731(methotrexate gamma-hydroxamic acid | CHEMBL244883)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant MMP7More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed