Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 50018676
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198035([(R)-2-methyl-1-(3'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 0.810nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198039([(R)-1-(4'-fluoro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198030([(R)-1-(3'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM12072(CHEMBL202932 | (R)-[1-(4-Methoxybiphenyl-4-sulfony...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198031([(R)-1-(4'-isopropoxy-biphenyl-4-sulfonylamino)-2-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM12072(CHEMBL202932 | (R)-[1-(4-Methoxybiphenyl-4-sulfony...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198031([(R)-1-(4'-isopropoxy-biphenyl-4-sulfonylamino)-2-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198040([(R)-2-methyl-1-(4'-pyrrolidin-1-yl-biphenyl-4-sul...)
Affinity DataIC50: 2nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198037([(R)-1-(3'-fluoro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM12072(CHEMBL202932 | (R)-[1-(4-Methoxybiphenyl-4-sulfony...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198031([(R)-1-(4'-isopropoxy-biphenyl-4-sulfonylamino)-2-...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198040([(R)-2-methyl-1-(4'-pyrrolidin-1-yl-biphenyl-4-sul...)
Affinity DataIC50: 5nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM12072(CHEMBL202932 | (R)-[1-(4-Methoxybiphenyl-4-sulfony...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50084293((S)-2-(4'-chloro-biphenyl-4-sulfonylamino)-3-methy...)
Affinity DataIC50: 9nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50084301(2-(4'-Fluoro-biphenyl-4-sulfonylamino)-3-methyl-bu...)
Affinity DataIC50: 10nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50084293((S)-2-(4'-chloro-biphenyl-4-sulfonylamino)-3-methy...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198038([(R)-1-(4'-ethoxy-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 12nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198039([(R)-1-(4'-fluoro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 13nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198035([(R)-2-methyl-1-(3'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 15nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198039([(R)-1-(4'-fluoro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198031([(R)-1-(4'-isopropoxy-biphenyl-4-sulfonylamino)-2-...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant MMP9 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198030([(R)-1-(3'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 24nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198035([(R)-2-methyl-1-(3'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198035([(R)-2-methyl-1-(3'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 26nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 28nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198030([(R)-1-(3'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198039([(R)-1-(4'-fluoro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 32nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198031([(R)-1-(4'-isopropoxy-biphenyl-4-sulfonylamino)-2-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50084301(2-(4'-Fluoro-biphenyl-4-sulfonylamino)-3-methyl-bu...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant MMP2 expressed in mouse myeloma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50084301(2-(4'-Fluoro-biphenyl-4-sulfonylamino)-3-methyl-bu...)
Affinity DataIC50: 43nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 45nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198033([(R)-2-methyl-1-(4'-methyl-biphenyl-4-sulfonylamin...)
Affinity DataIC50: 45nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-14(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50198034([(R)-1-(4'-chloro-biphenyl-4-sulfonylamino)-2-meth...)
Affinity DataIC50: 47nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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