Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50018551
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196941(N2-(2-chlorobenzyl)-N4-((3-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 3nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196932(N2-(2-(methylthio)benzyl)-N4-((4-(aminomethyl)cycl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196957(N2-(2-bromobenzyl)-N4-((4-(aminomethyl)cyclohexyl)...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196961(N2-(2-(trifluoromethylthio)benzyl)-N4-((4-(aminome...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196936(N2-(2,5-dichlorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 7nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196978(N2-(2,3-dichlorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196959(N2-(2-nitrobenzyl)-N4-((4-(aminomethyl)cyclohexyl)...)
Affinity DataIC50: 11nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196951(N2-(2-(trifluoromethyl)benzyl)-N4-((4-(aminomethyl...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196987(N2-(2,3-dimethylbenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 13nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196991(N2-(2-(difluoromethyl)benzyl)-N4-((4-(aminomethyl)...)
Affinity DataIC50: 15nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196952(N2-(2-methoxybenzyl)-N4-((4-(aminomethyl)cyclohexy...)
Affinity DataIC50: 17nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196972(N2-(2-(trifluoromethoxy)benzyl)-N4-((4-(aminomethy...)
Affinity DataIC50: 18nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196958(N2-(2-chlorobenzyl)-N4-(((1s,4s)-4-(aminomethyl)cy...)
Affinity DataIC50: 18nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196975(N2-(2,3-difluorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 22nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196990(N2-(2,4-dichlorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 27nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196982(N2-(2-chlorobenzyl)-N4-(((1r,4r)-4-(aminomethyl)cy...)
Affinity DataIC50: 29nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196980(N4-((4-(aminomethyl)cyclohexyl)methyl)-N2-(2,3-dih...)
Affinity DataIC50: 31nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196948(N*4*-(4-aminomethyl-cyclohexylmethyl)-N*2*-(2-meth...)
Affinity DataIC50: 34nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196956(N2-(2,5-difluorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 35nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196973(N*4*-(4-aminomethyl-cyclohexylmethyl)-N*2*-(3-meth...)
Affinity DataIC50: 39nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196954(N*4*-(4-aminomethyl-cyclohexylmethyl)-N*2*-bipheny...)
Affinity DataIC50: 39nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196935(N2-(2,6-difluorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 42nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196984(N2-(3-chloro-2-methylbenzyl)-N4-((4-(aminomethyl)c...)
Affinity DataIC50: 46nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196930(N2-(2-chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 46nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196985(N2-(2-fluorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 48nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196931(N2-(2-chlorobenzyl)-N4-((4-((dimethylamino)methyl)...)
Affinity DataIC50: 54nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196937(N2-(3-fluorophenethyl)-N4-((4-(aminomethyl)cyclohe...)
Affinity DataIC50: 54nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196965(N4-((4-(aminomethyl)cyclohexyl)methyl)-N2-(3-chlor...)
Affinity DataIC50: 60nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196968(N2-(4-fluorophenethyl)-N4-((4-(aminomethyl)cyclohe...)
Affinity DataIC50: 77nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196944(N2-(3-fluorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 83nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196934(N2-(3-chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 85nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196943(N2-(2-chlorobenzyl)-5-nitro-N4-(piperidin-4-ylmeth...)
Affinity DataIC50: 90nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196942(N4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-...)
Affinity DataIC50: 90nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196963(N4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-...)
Affinity DataIC50: 94nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196974(N2-(2,4-difluorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 100nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196966(N2-(2-chlorobenzyl)-N4-(7-aminoheptyl)-5-nitropyri...)
Affinity DataIC50: 110nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196977(N2-(2-fluorophenethyl)-N4-((4-(aminomethyl)cyclohe...)
Affinity DataIC50: 130nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196962(N2-(2-chlorobenzyl)-N4-(4-(aminomethyl)benzyl)-5-n...)
Affinity DataIC50: 160nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196945(N2-(4-chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 170nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196955(N*4*-(4-aminomethyl-cyclohexylmethyl)-5-nitro-N*2*...)
Affinity DataIC50: 180nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196983(N2-(2-chlorobenzyl)-N4-(3-(aminomethyl)benzyl)-5-n...)
Affinity DataIC50: 200nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196967(N2-(4-fluorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 210nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196971(N2-(3-methoxybenzyl)-N4-((4-(aminomethyl)cyclohexy...)
Affinity DataIC50: 210nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196933(N4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-...)
Affinity DataIC50: 270nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196930(N2-(2-chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 290nMAssay Description:Inhibition of PKCtheta in presence of 50 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196949(N2-(3,5-dichlorobenzyl)-N4-((4-(aminomethyl)cycloh...)
Affinity DataIC50: 400nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196981(N2-(2-chlorobenzyl)-N4-(5-aminopentyl)-5-nitropyri...)
Affinity DataIC50: 450nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196946((R)-N4-((4-(aminomethyl)cyclohexyl)methyl)-N2-(2,3...)
Affinity DataIC50: 460nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196960(N4-((4-(aminomethyl)cyclohexyl)methyl)-N2-benzyl-5...)
Affinity DataIC50: 500nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196930(N2-(2-chlorobenzyl)-N4-((4-(aminomethyl)cyclohexyl...)
Affinity DataIC50: 630nMAssay Description:Inhibition of PKCtheta in presence of 100 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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