Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50018442
TargetTranscription factor p65(Human)
Mediquest Therapeutics

Curated by ChEMBL
LigandPNGBDBM50195806(N-(3-(4-(3-aminopropylamino)butylamino)propyl)hexa...)
Affinity DataIC50: 230nMAssay Description:Inhibition of NF-kappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor p65(Human)
Mediquest Therapeutics

Curated by ChEMBL
LigandPNGBDBM50195808(N-(3-(4-(3-aminopropylamino)butylamino)propyl)deca...)
Affinity DataIC50: 310nMAssay Description:Inhibition of NF-kappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor p65(Human)
Mediquest Therapeutics

Curated by ChEMBL
LigandPNGBDBM50195809(N-(3-(4-(3-aminopropylamino)butylamino)propyl)dode...)
Affinity DataIC50: 340nMAssay Description:Inhibition of NF-kappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor p65(Human)
Mediquest Therapeutics

Curated by ChEMBL
LigandPNGBDBM50195807(N1-octadecanylsulfonyl-1,14-diamino-5,10-diazabuta...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of NF-kappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed