Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50018431
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  2nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195713(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  900nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)
Affinity DataEC50:  115nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  7nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  70nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  78nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  2nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  28nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  35nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataEC50:  2.65E+3nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50195712(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  2.80E+3nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  8nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  19nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195713(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  4nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195709(3-(2-((3-benzylureido)methyl)-4-(2-(5-methyl-2-phe...)
Affinity DataEC50:  2.68E+3nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195707(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  2.94E+3nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195707(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  527nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  198nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)
Affinity DataEC50:  515nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195712(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  1.02E+3nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataEC50:  986nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  308nMAssay Description:Activity at human PPARgamma in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  845nMAssay Description:Activity at human PPARalpha in CV1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195713(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195711(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 53nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195707(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 72nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)
Affinity DataIC50: 91nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195714(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 146nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195712(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 161nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195710(3-(2-((benzyloxycarbonyl)methyl)-4-(2-(5-methyl-2-...)
Affinity DataIC50: 441nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195716(3-{4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 449nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195715(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 516nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195709(3-(2-((3-benzylureido)methyl)-4-(2-(5-methyl-2-phe...)
Affinity DataIC50: 706nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195708(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195707(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 3.39E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 3.49E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195712(3-(4-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 4.96E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195713(3-(2-((isopropoxycarbonyl)methyl)-4-(2-(5-methyl-2...)
Affinity DataIC50: 9.94E+3nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50195709(3-(2-((3-benzylureido)methyl)-4-(2-(5-methyl-2-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-propyl-(5-pyridin-2yl-thiophene-2-sulfonyl)-amino]-pro-pyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from hPPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed