Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50037823
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  845nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  657nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195704(3-(2-(isobutoxycarbonyl)-5-(2-(5-methyl-2-phenylox...)
Affinity DataEC50:  8nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195705(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  9nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50195704(3-(2-(isobutoxycarbonyl)-5-(2-(5-methyl-2-phenylox...)
Affinity DataEC50:  1.72E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  2.75E+3nMAssay Description:Activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  2.39E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195706(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(p...)
Affinity DataEC50:  561nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  3.02E+3nMAssay Description:Activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataEC50:  19nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataEC50:  3nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  2.78E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085044(2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phen...)
Affinity DataEC50:  5nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataEC50:  77nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195706(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(p...)
Affinity DataEC50:  12nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  2.24E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085044(2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phen...)
Affinity DataEC50:  345nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195706(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(p...)
Affinity DataIC50: 11nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195704(3-(2-(isobutoxycarbonyl)-5-(2-(5-methyl-2-phenylox...)
Affinity DataIC50: 17nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195699(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataIC50: 21nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 24nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085044(2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phen...)
Affinity DataIC50: 25nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195705(5-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-ethoxy...)
Affinity DataIC50: 33nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 47nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 48nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085044(2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phen...)
Affinity DataIC50: 1.22E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataIC50: 1.29E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195704(3-(2-(isobutoxycarbonyl)-5-(2-(5-methyl-2-phenylox...)
Affinity DataIC50: 3.42E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195702(3-[4-[2-(2-biphenyl-4-yl-5-methyl-oxazol-4-yl)-eth...)
Affinity DataIC50: 3.49E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195706(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-(p...)
Affinity DataIC50: 4.68E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM50195703(3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)-2-((...)
Affinity DataIC50: 8.40E+3nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tritium labeled ligand from human PPARalpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tritium labeled ligand from human PPARgamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)