Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50037781
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195511(N-(4'-methylcyclohexyl)-1-(o-fluorobenzyl)-7-methy...)
Affinity DataEC50:  138nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataEC50:  204nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195516(N-(4'-methylcyclohexyl)-1-(p-fluorobenzyl)-7-methy...)
Affinity DataEC50:  27nMAssay Description:Activity at CB1 receptor assessed as stimulation of [35S]GTP-gamma-S binding in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195527(N-cycloheptyl-1-(p-fluorobenzyl)-7-methyl-1,8-naph...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195516(N-(4'-methylcyclohexyl)-1-(p-fluorobenzyl)-7-methy...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195513(N-cyclohexyl-7-chloro-1-(2-morpholin-4-ylethyl)-qu...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50072769(N-(2-chloroethyl)icosa-5,8,11,14-tetraenamide | (5...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195527(N-cycloheptyl-1-(p-fluorobenzyl)-7-methyl-1,8-naph...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195517(N-cyclohexyl-1-benzylquinolin-4(1H)-on-3-carboxami...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195514(N-cycloheptyl-1-benzyl-7-methyl-1,8-naphthyridin-4...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195511(N-(4'-methylcyclohexyl)-1-(o-fluorobenzyl)-7-methy...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195516(N-(4'-methylcyclohexyl)-1-(p-fluorobenzyl)-7-methy...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195519(N-cyclohexyl-7-methyl-1-benzyl-1,8-naphthyridin-4(...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195529(N-cyclohexyl-1-(p-fluorbenzyl)-1,8-naphthyridin-4(...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195518(N-cycloheptyl-1-(o-fluorbenzyl)-7-methyl-1,8-napht...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195528(N-cyclohexyl-7-methyl-1-phenethyl-1,8-naphthyridin...)
Affinity DataKi:  16.3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195525(N-cyclohexyl-7-chloro-1-(o-fluorbenzyl)-1,8-naphth...)
Affinity DataKi:  18.1nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195515(N-cyclohexyl-7-chloro-1-(p-fluorbenzyl)-1,8-naphth...)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195522(N-cyclohexyl-1-benzyl-7-chloro-1,8-naphthyridin-4(...)
Affinity DataKi:  24.6nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195523(N-cyclohexyl-7-methyl-1-(4-methoxybenzyl)-1,8-naph...)
Affinity DataKi:  35.8nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195511(N-(4'-methylcyclohexyl)-1-(o-fluorobenzyl)-7-methy...)
Affinity DataKi:  37.5nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195524(N-(4'-methylcyclohexyl)-7-chloro-1-(2-morpholin-4-...)
Affinity DataKi:  40.5nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195520(N-cyclohexyl-1-benzyl-1,8-naphthyridin-4(1H)-on-3-...)
Affinity DataKi:  48.6nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195526(N-cyclopentyl-7-methyl-1-(2-morpholin-4-ylethyl)-1...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195512(N-cyclohexyl-1-(2-morpholin-4-yl-ethyl)-1,8-naphth...)
Affinity DataKi:  67.2nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50072769(N-(2-chloroethyl)icosa-5,8,11,14-tetraenamide | (5...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195519(N-cyclohexyl-7-methyl-1-benzyl-1,8-naphthyridin-4(...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195514(N-cycloheptyl-1-benzyl-7-methyl-1,8-naphthyridin-4...)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195518(N-cycloheptyl-1-(o-fluorbenzyl)-7-methyl-1,8-napht...)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195525(N-cyclohexyl-7-chloro-1-(o-fluorbenzyl)-1,8-naphth...)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195529(N-cyclohexyl-1-(p-fluorbenzyl)-1,8-naphthyridin-4(...)
Affinity DataKi:  384nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  458nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195522(N-cyclohexyl-1-benzyl-7-chloro-1,8-naphthyridin-4(...)
Affinity DataKi:  464nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195515(N-cyclohexyl-7-chloro-1-(p-fluorbenzyl)-1,8-naphth...)
Affinity DataKi:  495nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195508(N-cyclohexyl-7-methyl-1-[2-(4-phenylpiperazin-1-yl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195513(N-cyclohexyl-7-chloro-1-(2-morpholin-4-ylethyl)-qu...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195509(4-hydroxy-N-(4-methylcyclohexyl)-1-(2-morpholin-4-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195521(N-cyclohexyl-1-benzyl-4-hydroxy-7-methyl-1,2,3,4-t...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195510(N-cyclohexyl-1-(o-fluorbenzyl)-4-hydroxy-7-methyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195512(N-cyclohexyl-1-(2-morpholin-4-yl-ethyl)-1,8-naphth...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195509(4-hydroxy-N-(4-methylcyclohexyl)-1-(2-morpholin-4-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195517(N-cyclohexyl-1-benzylquinolin-4(1H)-on-3-carboxami...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195521(N-cyclohexyl-1-benzyl-4-hydroxy-7-methyl-1,2,3,4-t...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195526(N-cyclopentyl-7-methyl-1-(2-morpholin-4-ylethyl)-1...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195528(N-cyclohexyl-7-methyl-1-phenethyl-1,8-naphthyridin...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195523(N-cyclohexyl-7-methyl-1-(4-methoxybenzyl)-1,8-naph...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195520(N-cyclohexyl-1-benzyl-1,8-naphthyridin-4(1H)-on-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in DBA/J2 mouse brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195510(N-cyclohexyl-1-(o-fluorbenzyl)-4-hydroxy-7-methyl-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50195508(N-cyclohexyl-7-methyl-1-[2-(4-phenylpiperazin-1-yl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in DBA/J2 mouse spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2012
Entry Details Article
PubMed
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