Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50018377
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  882nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195082(2-((5-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  105nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195080(2-((5-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195081(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195087(2-ethoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195078(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyra...)
Affinity DataEC50:  1.89E+3nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195084(2-((5-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  867nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195086(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195083((R)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195075(2-ethoxy-3-(5-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataEC50:  886nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195075(2-ethoxy-3-(5-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataEC50:  887nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195076(2-methoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataEC50:  3.14E+3nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195076(2-methoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195086(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  226nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195087(2-ethoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195083((R)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195084(2-((5-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195074(2-((5-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  1.57E+3nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195085(2-((2-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  335nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195082(2-((5-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  437nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195074(2-((5-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195078(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyra...)
Affinity DataEC50:  156nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195081(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195080(2-((5-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195085(2-((2-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195074(2-((5-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  20nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  43nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195084(2-((5-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  43nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195087(2-ethoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)eth...)
Affinity DataKi:  73nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195082(2-((5-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  93nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195080(2-((5-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  150nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195078(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyra...)
Affinity DataKi:  160nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195086(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  210nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195080(2-((5-(2-(2-(4-chlorophenyl)-5-methyloxazol-4-yl)e...)
Affinity DataKi:  300nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195079((S)-2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)...)
Affinity DataKi:  340nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195076(2-methoxy-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)et...)
Affinity DataKi:  348nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataKi:  440nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195082(2-((5-(2-(2-(4-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  840nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195075(2-ethoxy-3-(5-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataKi:  840nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195075(2-ethoxy-3-(5-(3-(5-methyl-2-phenyloxazol-4-yl)pro...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195084(2-((5-(2-(5-methyl-2-m-tolyloxazol-4-yl)ethoxy)pyr...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195081(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195074(2-((5-(2-(2-(3-methoxyphenyl)-5-methyloxazol-4-yl)...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195086(2-((5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyri...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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