Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50037815
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194351(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194342(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194331(2-hydroxy-2-(5-(2,2,2-trifluoroacetamido)-6-(trifl...)
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194352(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194350(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 180nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194337(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 180nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194330(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194353(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-2-h...)
Affinity DataIC50: 440nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194326(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194345(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194340(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 460nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194327(2-(5-cyano-6-(trifluoromethyl)-1H-indol-2-yl)-2-hy...)
Affinity DataIC50: 480nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194354(2-(5-chloro-1H-indol-2-yl)-1-(4-chlorophenylthio)p...)
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194344(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 720nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194346(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 820nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194328(1-(4-aminophenylthio)-2-(5-chloro-6-(trifluorometh...)
Affinity DataIC50: 930nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194339(biphenyl-4-carboxylic acid 2-hydroxy-2-(5-nitro-6-...)
Affinity DataIC50: 940nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194335(1-(3,4-dichlorophenylthio)-2-(5-nitro-6-(trifluoro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194355(2-(5-cyano-6-(trifluoromethyl)-1H-indol-2-yl)-2-hy...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194348(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194347(2-(1-(4-chlorophenylthio)-2-hydroxypropan-2-yl)-6-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194332(2-(1-(4-fluorophenylthio)-2-hydroxypropan-2-yl)-6-...)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194349(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194333(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194341(2-(2-hydroxy-1-(phenylthio)propan-2-yl)-6-(trifluo...)
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194329(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194338(2-(5-amino-6-(trifluoromethyl)-1H-indol-2-yl)-2-hy...)
Affinity DataIC50: 4.10E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194336(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 4.90E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194336(2-(5-chloro-6-(trifluoromethyl)-1H-indol-2-yl)-1-(...)
Affinity DataIC50: 5.10E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194334(2-hydroxy-2-(5-nitro-6-(trifluoromethyl)-1H-indol-...)
Affinity DataIC50: 6.40E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
Johnson and Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50194343(2-(1-(4-fluorophenylsulfonyl)-2-hydroxypropan-2-yl...)
Affinity DataIC50: 6.90E+3nMAssay Description:Displacement of [3H]R1881 from rat androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed