Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50018253
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >1.94E+3nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >7.03E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >9.46E+3nMAssay Description:Activity at human LPA2 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193515(1-fluoro-(3S)-hydroxyl-4-oleoyloxylbutane 1,3-cycl...)
Affinity DataIC50: 106nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193518(3-hydroxyl-4-palmitoyloxylbutane 1,3-cyclic phosph...)
Affinity DataIC50: 799nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193517(3-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphono...)
Affinity DataIC50: 941nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193517(3-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphono...)
Affinity DataIC50: 1.27E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193518(3-hydroxyl-4-palmitoyloxylbutane 1,3-cyclic phosph...)
Affinity DataIC50: 2.34E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193515(1-fluoro-(3S)-hydroxyl-4-oleoyloxylbutane 1,3-cycl...)
Affinity DataIC50: 7.72E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193515(1-fluoro-(3S)-hydroxyl-4-oleoyloxylbutane 1,3-cycl...)
Affinity DataKi:  60.7nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193518(3-hydroxyl-4-palmitoyloxylbutane 1,3-cyclic phosph...)
Affinity DataKi:  314nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193517(3-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphono...)
Affinity DataKi:  403nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193517(3-hydroxyl-4-oleoyloxylbutane 1,3-cyclic phosphono...)
Affinity DataKi:  636nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193518(3-hydroxyl-4-palmitoyloxylbutane 1,3-cyclic phosph...)
Affinity DataKi:  1.15E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
The University of Utah

Curated by ChEMBL
LigandPNGBDBM50193515(1-fluoro-(3S)-hydroxyl-4-oleoyloxylbutane 1,3-cycl...)
Affinity DataKi:  3.17E+3nMAssay Description:Activity at human LPA3 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed