Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50018058
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190601((2S,4R,5R)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190607((2S,4R,5R)-2-benzhydryl-5-(benzylamino)-tetrahydro...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190605(cis-(3S-6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  6.60nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  8.60nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190606((2S,4R,5R)-2-benzhydryl-5-(4-hydroxy-benzylamino)-...)
Affinity DataKi:  10nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  11nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190600(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  12nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190610((2R,4S,5S)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  13nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190608(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  13nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190605(cis-(3S-6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  15nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190601((2S,4R,5R)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  15nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190600(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  16nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  16nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190608(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  16nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190611(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  20nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  26nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190598(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  26nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190611(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  35nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  38nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190611(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  38nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190602(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  41nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190598(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  44nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190598(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  46nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190611(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  54nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190604(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  60nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190608(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  62nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190604(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  65nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190604(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  65nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190602(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  67nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190604(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  82nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  85nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  91nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190599((2R,4S, 5S)-2-benzhydryl-5-(4-hydroxy-benzylamino)...)
Affinity DataKi:  92nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190599((2R,4S, 5S)-2-benzhydryl-5-(4-hydroxy-benzylamino)...)
Affinity DataKi:  94nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM22165(Vanoxerine | CHEMBL542933 | GBR-12909 | CHEMBL5438...)
Affinity DataKi:  102nMAssay Description:Inhibition of NET-mediated [3H]NE uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190602(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  114nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  115nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190598(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  118nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190601((2S,4R,5R)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  120nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190599((2R,4S, 5S)-2-benzhydryl-5-(4-hydroxy-benzylamino)...)
Affinity DataKi:  125nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190608(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  142nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190600(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  142nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190606((2S,4R,5R)-2-benzhydryl-5-(4-hydroxy-benzylamino)-...)
Affinity DataKi:  172nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190609((2S,4R,5R)-5-(4-methoxybenzylamino)-2-benzhydryl-t...)
Affinity DataKi:  183nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190610((2R,4S,5S)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  184nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190602(cis-(3R,6R)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  187nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190605(cis-(3S-6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(1...)
Affinity DataKi:  214nMAssay Description:Inhibition of DAT-mediated [3H]DA uptake in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190610((2R,4S,5S)-2-benzhydryl-5-[(1H-indol-5-ylmethyl)-a...)
Affinity DataKi:  223nMAssay Description:Inhibition of SERT-mediated [3H]5-HT uptake in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50190603(cis-(3S,6S)-(6-benzhydryl-tetrahydropyran-3-yl)-(4...)
Affinity DataKi:  226nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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