Compile Data Set for Download or QSAR
Report error Found 155 Enz. Inhib. hit(s) with all data for entry = 50037726
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189842(2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo...)
Affinity DataEC50:  2.60nMAssay Description:Activity at human D4.4 receptor expressed in CHOK1 cells assessed as stimulation of [35S]GTP-gammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataEC50:  1.40nMAssay Description:Activity at human D4.2 receptor assessed as [3H]thymidine incorporation in CHO 10001 cells by mitogenesis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189842(2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo...)
Affinity DataEC50:  1.80nMAssay Description:Activity at human D4.2 receptor assessed as [3H]thymidine incorporation in CHO 10001 cells by mitogenesis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataEC50:  4.5nMAssay Description:Activity at human D4.4 receptor expressed in CHOK1 cells assessed as stimulation of [35S]GTP-gammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataEC50:  3nMAssay Description:Activity at human D4.2 receptor assessed as [3H]thymidine incorporation in CHO 10001 cells by mitogenesis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataEC50:  0.520nMAssay Description:Activity at human D4.2 receptor assessed as [3H]thymidine incorporation in CHO 10001 cells by mitogenesis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM84637(NSC_54562 | CHEMBL240773 | QUINPIROLE | CAS_85760-...)
Affinity DataEC50:  49nMAssay Description:Activity at human D4.4 receptor expressed in CHOK1 cells assessed as stimulation of [35S]GTP-gammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50094505(2-(4-Phenyl-piperazin-1-ylmethyl)-1H-indole-5-carb...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189852(8-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189843(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  0.940nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189839(6-bromo-2-[4-(3,4-dichlorophenyl)piperazin-1-ylmet...)
Affinity DataKi:  0.990nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189851(8-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.990nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50094503(2-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-in...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189856(6-chloro-2-[4-(3,4-dichlorophenyl)piperazin-1-ylme...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189853(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189848(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imid...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189840(6-chloro-2-[4-(2-methoxyphenyl)piperazin-1-ylmethy...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189847(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189849(6-chloro-2-[4-(4-chlorophenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189857(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50073805(FAUC 113 | 3-[4-(4-Chloro-phenyl)-piperazin-1-ylme...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189846(6-chloro-2-[4-(4-fluorophenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189842(2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189840(6-chloro-2-[4-(2-methoxyphenyl)piperazin-1-ylmethy...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in porcine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189843(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189837(2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189843(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189840(6-chloro-2-[4-(2-methoxyphenyl)piperazin-1-ylmethy...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189852(8-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189840(6-chloro-2-[4-(2-methoxyphenyl)piperazin-1-ylmethy...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189852(8-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189857(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189855(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]-6-(...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189851(8-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189857(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189851(8-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189844(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-5-(pyr...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of Tours

Curated by ChEMBL
LigandPNGBDBM50189847(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]-6-meth...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
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