Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50017971
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189380(N-(2-(4-benzylpiperidine-1-carbonyl)-1H-benzo[d]im...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189391((5-hydroxy-1H-benzo[d]imidazol-2-yl)(4-(p-tolyloxy...)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189383((4-(3-methoxybenzyl)piperidin-1-yl)(5-hydroxy-1H-b...)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50204862(N-[2-(4-Benzyl-piperidin-1-ylmethyl)-3H-benzoimida...)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50204884(6-(2-(4-(4-fluorobenzyl)piperidin-1-yl)ethylsulfin...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189385((4-(4-fluorobenzyl)piperidin-1-yl)(5-hydroxy-1H-be...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50241126((4-benzylpiperidin-1-yl)(5-hydroxy-1H-benzo[d]imid...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50241129((5-hydroxy-1H-benzoimidazol-2-yl)-[4-(4-methyl-ben...)
Affinity DataIC50: 4.40nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50241127((5-hydroxy-1H-benzoimidazol-2-yl)-[4-(3-methyl-ben...)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50241128((4-(3-fluorobenzyl)piperidin-1-yl)(5-hydroxy-1H-be...)
Affinity DataIC50: 5.20nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189388((4-(4-fluorophenoxy)piperidin-1-yl)(5-hydroxy-1H-b...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50080029(CHEMBL305195 | 4-[(1R,2S)-3-(4-Benzyl-piperidin-1-...)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189384((5-hydroxy-1H-benzoimidazol-2-yl)-[4-(2-methyl-ben...)
Affinity DataIC50: 8.40nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189389((4-benzylpiperidin-1-yl)(4-hydroxy-1H-benzo[d]imid...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50134651((4-Benzyl-piperidin-1-yl)-(6-hydroxy-1H-indol-2-yl...)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189387((4-(4-chlorophenoxy)piperidin-1-yl)(5-hydroxy-1H-b...)
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50189390((5-amino-1H-benzo[d]imidazol-2-yl)(4-benzylpiperid...)
Affinity DataIC50: 143nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50080016((E)-1-(4-Benzyl-piperidin-1-yl)-3-(4-hydroxy-pheny...)
Affinity DataIC50: 196nMAssay Description:Displacement of [3H]Ro25-6981 from NR2B NMDA receptor in rat forebrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed