Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50017928
TargetDelta-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(H-Dmt-Tic-Glu-Dap(6DMN)-NH(2) | CHEMBL208916)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataKi:  41.3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(H-Dmt-Tic-Glu-Dap(6DMN)-NH(2) | CHEMBL208916)
Affinity DataIC50: 100nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S)-NH-fluorescei...)
Affinity DataIC50: 120nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S)-NH-fluorescei...)
Affinity DataIC50: 200nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataIC50: 244nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-Dap(6DMN)-NH2 | ...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S)-NH-fluorescei...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-Dap(6DMN)-NH2 | ...)
Affinity DataIC50: 253nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-Dap(6DMN)-NH2 | ...)
Affinity DataIC50: 300nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(H-Tyr-Pro-Dap(6DMN)-Phe-NH2 | CHEMBL207661)
Affinity DataIC50: 389nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(H-Tyr-Pro-Dap(6DMN)-Phe-NH2 | CHEMBL207661)
Affinity DataIC50: 500nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S)-NH-fluorescei...)
Affinity DataKi:  668nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(H-Tyr-Pro-Dap(6DMN)-Phe-NH2 | CHEMBL207661)
Affinity DataKi:  839nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(H-Tyr-Pro-Dap(6DMN)-Phe-NH2 | CHEMBL207661)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-Dap(6DMN)-NH2 | ...)
Affinity DataKi:  5.94E+3nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(H-Dmt-Tic-Glu-Dap(6DMN)-NH(2) | CHEMBL208916)
Affinity DataKi:  7.88E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed