Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50000586
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007538(CHEMBL25626 | 8-(2-Azetidin-1-yl-ethyl)-3-chloro-6...)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of [3H]mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007542(CHEMBL24835 | 3-Chloro-8-(2-dimethylamino-ethyl)-6...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007536(CHEMBL24517 | [3-(5-Chloro-pyridin-2-yl)-3-pyridin...)
Affinity DataIC50: 24nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007539(CHEMBL24031 | 8-(2-Dimethylamino-ethyl)-6-methyl-7...)
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007540(CHEMBL279907 | [3-(4-Chloro-phenyl)-3-(5-chloro-py...)
Affinity DataIC50: 430nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007535(CHEMBL25198 | 8-(2-Azetidin-1-yl-ethyl)-3-chloro-6...)
Affinity DataIC50: 870nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007541(CHEMBL283760 | 3-Chloro-8-(2-dimethylamino-ethyl)-...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
A.H. Robins

Curated by ChEMBL
LigandPNGBDBM50007537(CHEMBL25622 | 8-(2-Dimethylamino-ethyl)-6-methyl-7...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of [3H]mepyramine binding to the Histamine H1 receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed