Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50017796
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186608(3-((4-hydroxy-3,5-dimethoxy)phenyl)prop-1,2-diyl d...)
Affinity DataEC50:  4.90E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186604(4-((N-(3-(3,5-di-tert-butyl-4-hydroxyphenyl)propyl...)
Affinity DataEC50:  410nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156307(4-(3-Nitrooxy-propyl)-phenol | 3-(4-hydroxyphenyl)...)
Affinity DataEC50:  1.00E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156305(2,5,7,8-Tetramethyl-2-(3-nitrooxy-propoxymethyl)-c...)
Affinity DataEC50:  1.20E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186613(4-hydroxymethyl-2-oxy-furazan-3-carboxylic acid am...)
Affinity DataEC50:  6.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156310(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)phen...)
Affinity DataEC50:  12nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186612(1,2-bis-nitrooxy-propane | CHEMBL206527)
Affinity DataEC50:  240nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186606(3-(4-hydroxyphenyl)prop-1,2-diyl dinitrate | CHEMB...)
Affinity DataEC50:  130nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156310(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)phen...)
Affinity DataEC50:  360nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186608(3-((4-hydroxy-3,5-dimethoxy)phenyl)prop-1,2-diyl d...)
Affinity DataEC50:  640nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186611(3-(4-hydroxy-3,5-dimethoxyphenyl)propyl nitrate | ...)
Affinity DataEC50:  4.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186610(3-((4-hydroxy-3,5-di-tert-butyl)phenyl)prop-1,2-di...)
Affinity DataEC50:  3.30E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186605(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)-2,6...)
Affinity DataEC50:  500nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186603(4-((N-((6-hydroxy-2,5,7,8-tetramethylchroman-2-yl)...)
Affinity DataEC50:  1.90E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156303(2-(4-Benzenesulfonyl-5-oxy-furazan-3-yloxymethyl)-...)
Affinity DataEC50:  670nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186607(4-dimethylaminomethyl-2-oxy-furazan-3-carboxylic a...)
Affinity DataEC50:  3.10E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186603(4-((N-((6-hydroxy-2,5,7,8-tetramethylchroman-2-yl)...)
Affinity DataEC50:  1.50E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156303(2-(4-Benzenesulfonyl-5-oxy-furazan-3-yloxymethyl)-...)
Affinity DataEC50:  44nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156308(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)-2,6...)
Affinity DataEC50:  4.80E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156309(2,6-Di-tert-butyl-4-(3-nitrooxy-propyl)-phenol | 3...)
Affinity DataEC50:  4.00E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156304(4-ethoxy-3-(phenylsulfonyl)-1,2,5-oxadiazole 2-oxi...)
Affinity DataEC50:  12nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186606(3-(4-hydroxyphenyl)prop-1,2-diyl dinitrate | CHEMB...)
Affinity DataEC50:  6.50E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186605(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)-2,6...)
Affinity DataEC50:  22nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156306(1-nitrooxy-propane | CHEMBL188554)
Affinity DataEC50:  4.10E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50186604(4-((N-(3-(3,5-di-tert-butyl-4-hydroxyphenyl)propyl...)
Affinity DataEC50:  7.40E+3nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156305(2,5,7,8-Tetramethyl-2-(3-nitrooxy-propoxymethyl)-c...)
Affinity DataEC50:  1.00E+4nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic strips in presence of 1 uM ODQMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50156308(4-(3-(3-benzenesulfonylfuroxan-4-yloxy)propyl)-2,6...)
Affinity DataEC50:  110nMAssay Description:Vasodilator activity assessed as ability to relax phenylephrine-induced contraction of Wistar rat aortic stripsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed