Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50037684
LigandPNGBDBM50185264(N-((1H-pyrrol-3-yl)methyl)-2-(5-nitro-1H-indol-3-y...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50370710(CHEMBL1162923)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185269(N-(furan-3-ylmethyl)-2-(5-nitro-1H-indol-3-yl)-2-o...)
Affinity DataKi:  56.6nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185273(N-((1H-pyrrol-2-yl)methyl)-2-(5-nitro-1H-indol-3-y...)
Affinity DataKi:  73.5nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185264(N-((1H-pyrrol-3-yl)methyl)-2-(5-nitro-1H-indol-3-y...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50370710(CHEMBL1162923)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185269(N-(furan-3-ylmethyl)-2-(5-nitro-1H-indol-3-yl)-2-o...)
Affinity DataKi:  236nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185266(N-((1H-pyrrol-2-yl)methyl)-2-(1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  271nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185277(N-((1H-pyrrol-3-yl)methyl)-2-(1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  272nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha1 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185273(N-((1H-pyrrol-2-yl)methyl)-2-(5-nitro-1H-indol-3-y...)
Affinity DataKi:  585nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185277(N-((1H-pyrrol-3-yl)methyl)-2-(1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  681nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha5 receptor plus beta-3-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM26266(Ambien | CHEMBL911 | ZPM | N,N-dimethyl-2-[6-methy...)
Affinity DataKi:  765nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185266(N-((1H-pyrrol-2-yl)methyl)-2-(1H-indol-3-yl)-2-oxo...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha5 receptor plus beta-3-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50185264(N-((1H-pyrrol-3-yl)methyl)-2-(5-nitro-1H-indol-3-y...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha5 receptor plus beta-3-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed