Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017676
TargetCholecystokinin receptor type A(Human)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50185261(4-(3,4-dichlorobenzamido)-5-((3-methoxypropyl)(pen...)
Affinity DataIC50: 195nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50185262((+/-)-2-(2-(1H-indole-2-carboxamido)benzamido)-3-p...)
Affinity DataIC50: 197nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50185259(2(R,S)-{2-[(1H-indole-2-carbonyl)amino]-benzoylami...)
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50185260((+/-)-2-(2-cinnamamidobenzamido)-3-phenylpropanoic...)
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Human)
University of Naples Federico Ii

Curated by ChEMBL
LigandPNGBDBM50185263(2(R,S)-{2-[(2-acetylaminocinnamoyl)amino]benzoylam...)
Affinity DataIC50: 1.27E+4nMAssay Description:Displacement of [111In]DTPA-Glu-Gly-[Tyr27(SO3H)]-CCK8 from human CCK1 receptor in A431 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed