Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 50017593
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against hMC1R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.300nMAssay Description:Activity against hMC1R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL263822)
Affinity DataEC50:  1.20nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184355(c[Nle-Gln-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20431...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184355(c[Nle-Gln-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20431...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184361(c[Nle-Val-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL41357...)
Affinity DataIC50: 1.70nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  1.90nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184361(c[Nle-Val-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL41357...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184365(c[Nle-Arg-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20426...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184356(c[Nle-His-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL42559...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184365(c[Nle-Arg-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20426...)
Affinity DataIC50: 2.60nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  2.90nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  3.30nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20486...)
Affinity DataIC50: 3.80nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20486...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataIC50: 7.5nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184366(c[Nle-Pro-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20376...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184356(c[Nle-His-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL42559...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184366(c[Nle-Pro-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20376...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184361(c[Nle-Val-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL41357...)
Affinity DataEC50:  16nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20486...)
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184352(c[Nle-Val-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL427205)
Affinity DataEC50:  27nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184354(c[Nle-Glu-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL38325...)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184353(c[Nle-His-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL446185)
Affinity DataEC50:  37nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184354(c[Nle-Glu-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL38325...)
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184355(c[Nle-Gln-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20431...)
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL263822)
Affinity DataIC50: 68nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL380638)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184365(c[Nle-Arg-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20426...)
Affinity DataIC50: 77nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184356(c[Nle-His-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL42559...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184353(c[Nle-His-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL446185)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184352(c[Nle-Val-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL427205)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184355(c[Nle-Gln-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20431...)
Affinity DataEC50:  130nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184354(c[Nle-Glu-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL38325...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL263822)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184358(c[Nle-Asp-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL203170)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184353(c[Nle-His-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL446185)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184350(c[Nle-Asp-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL40914...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL263822)
Affinity DataEC50:  174nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184361(c[Nle-Val-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL41357...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184352(c[Nle-Val-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL427205)
Affinity DataEC50:  180nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184360(c[Nle-Nle-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL20486...)
Affinity DataEC50:  200nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184350(c[Nle-Asp-D-Nal(2')-Arg-Trp-Glu]-NH2 | CHEMBL40914...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against hMC5R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL380638)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184363(c[Nle-Arg-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL263822)
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184364(c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL203602)
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against hMC3R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184364(c[Nle-Gln-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL203602)
Affinity DataEC50:  300nMAssay Description:Activity against hMC5R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50184362(c[Nle-Nle-D-Phe-Arg-Trp-Glu]-NH2 | CHEMBL380638)
Affinity DataEC50:  300nMAssay Description:Activity against hMC3R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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