Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50017582
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184279(1-benzyl-3-(4-morpholinophenylamino)pyrrolidine-2,...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM32184(CHEMBL209511 | N-(4-chloro-2-hydroxyphenyl)benzene...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM55151(2-[2-[3,4-bis(oxidanyl)phenyl]-2-oxidanylidene-eth...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184280(N-(4-hydroxy-3-methylphenyl)-3-methoxybenzamide | ...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184276(3-(1-hydroxy-3,3-dimethyl-3,4,10,11-tetrahydro-2H-...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184282(4-methoxy-2-(3-(thiophen-2-yl)-1H-pyrazol-4-yl)phe...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184281(3-(4-fluorophenoxy)-7,8-dihydroxy-4H-chromen-4-one...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184283(1-(3-chlorophenyl)pyrazolidine-3,5-dione | CHEMBL2...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM32185(6-[5-(4-hydroxy-3-methoxyphenyl)-3-pyrazolidinylid...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184278(N-(4-(2-amino-4-methylthiazol-5-yl)thiazol-2-yl)py...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Hsp90 by recombinant ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM32185(6-[5-(4-hydroxy-3-methoxyphenyl)-3-pyrazolidinylid...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Her2 in SKBr3 cells by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM32184(CHEMBL209511 | N-(4-chloro-2-hydroxyphenyl)benzene...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of Her2 in SKBr3 cells by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
The University of Kansas

Curated by ChEMBL
LigandPNGBDBM50184276(3-(1-hydroxy-3,3-dimethyl-3,4,10,11-tetrahydro-2H-...)
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of Her2 in SKBr3 cells by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed