Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 50017443
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182237(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182221(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182245(N-((R)-6-((isobutylamino)methyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182230(2-((S)-1-(benzo[b]thiophen-3-ylsulfonyl)piperidin-...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182231(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182237(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182222(N-((R)-6-((cyclopropylmethylamino)methyl)-1,2,3,4-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182220(N-((R)-6-((2-methoxyethylamino)methyl)-1,2,3,4-tet...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182231(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182221(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182222(N-((R)-6-((cyclopropylmethylamino)methyl)-1,2,3,4-...)
Affinity DataIC50: 31nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182245(N-((R)-6-((isobutylamino)methyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182220(N-((R)-6-((2-methoxyethylamino)methyl)-1,2,3,4-tet...)
Affinity DataIC50: 46nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182232(N-((R)-6-((cyclopropylamino)methyl)-1,2,3,4-tetrah...)
Affinity DataIC50: 47nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182232(N-((R)-6-((cyclopropylamino)methyl)-1,2,3,4-tetrah...)
Affinity DataIC50: 48nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182234(N-((R)-6-((cyclobutylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182234(N-((R)-6-((cyclobutylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 58nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182229(N-((R)-6-((neopentylamino)methyl)-1,2,3,4-tetrahyd...)
Affinity DataIC50: 59nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182236(N-((R)-6-((dimethylamino)methyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 62nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182230(2-((S)-1-(benzo[b]thiophen-3-ylsulfonyl)piperidin-...)
Affinity DataIC50: 66nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182228(N-((R)-6-((isopropylamino)methyl)-1,2,3,4-tetrahyd...)
Affinity DataIC50: 72nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182241(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182239(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 93nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182225(N-((R)-7-((tert-butylamino)methyl)chroman-4-yl)-2-...)
Affinity DataIC50: 95nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182228(N-((R)-6-((isopropylamino)methyl)-1,2,3,4-tetrahyd...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182241(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182239(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182235(2-((S)-1-(benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)p...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182236(N-((R)-6-((dimethylamino)methyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182225(N-((R)-7-((tert-butylamino)methyl)chroman-4-yl)-2-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182235(2-((S)-1-(benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)p...)
Affinity DataIC50: 180nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182238(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182246(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182229(N-((R)-6-((neopentylamino)methyl)-1,2,3,4-tetrahyd...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182238(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182246(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182242(2-[(S)-1-(biphenyl-4-sulfonyl)-piperidin-2-yl]-N-[...)
Affinity DataIC50: 540nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182226(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182224(2-((S)-1-(4-butoxyphenylsulfonyl)piperidin-2-yl)-N...)
Affinity DataIC50: 590nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182247(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 610nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182242(2-[(S)-1-(biphenyl-4-sulfonyl)-piperidin-2-yl]-N-[...)
Affinity DataIC50: 690nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182227(N-((R)-6-((2,2,2-trifluoroethylamino)methyl)-1,2,3...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182223(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 780nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182226(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 810nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182240(N-((R)-7-((tert-butylamino)methyl)chroman-4-yl)-2-...)
Affinity DataIC50: 960nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182233(N-((R)-6-(azetidin-1-ylmethyl)-1,2,3,4-tetrahydron...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182224(2-((S)-1-(4-butoxyphenylsulfonyl)piperidin-2-yl)-N...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182223(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182240(N-((R)-7-((tert-butylamino)methyl)chroman-4-yl)-2-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50182243(N-((R)-6-((tert-butylamino)methyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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