Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50017261
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179827(2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propo...)
Affinity DataEC50:  110nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179823((S)-2-methyl-2-((4-(3-(8-methyl-2-oxo-4-(trifluoro...)
Affinity DataEC50:  10nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179835(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  20nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127933(CHEMBL1783044 | CHEMBL300026 | 5-(4-(3-(4-(4-fluor...)
Affinity DataEC50:  735nMAssay Description:Binding affinity to human PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179830((S)-2-(4-(3-(2-chloro-4-cyclohexylphenoxy)propoxy)...)
Affinity DataEC50:  1nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179838((S)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)p...)
Affinity DataEC50:  20nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179827(2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propo...)
Affinity DataEC50:  106nMAssay Description:Binding affinity to human PPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179836((S)-2-(4-(3-(2-chloro-4-(2,2,2-trifluoroethoxy)phe...)
Affinity DataEC50:  7.80nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179834(2-(3-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  2.23E+3nMAssay Description:Binding affinity to human PPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179843(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  454nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179819(2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butox...)
Affinity DataEC50:  284nMAssay Description:Transactivation by human PPAR delta in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179829(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  2.70nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179833((S)-2-(4-(3-(2-chloro-4-(trifluoromethyl)phenoxy)p...)
Affinity DataEC50:  2.90nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179824((S)-2-(4-(3-(2-chloro-4-(trifluoromethoxy)phenoxy)...)
Affinity DataEC50:  2.10nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179819(2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butox...)
Affinity DataEC50:  545nMAssay Description:Binding affinity to human PPAR deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179828((S)-2-((4-(3-(6-chloro-2-oxo-4-(trifluoromethyl)-2...)
Affinity DataEC50:  44nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179838((S)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)p...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR gamma in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179816((S)-2-(4-(3-(2-chloro-4-(4,4-dimethylcyclohexyl)ph...)
Affinity DataEC50:  27.5nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179819(2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butox...)
Affinity DataEC50:  35nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179821((S)-2-(4-(3-(2-chlorophenoxy)propoxy)benzyl)-2-met...)
Affinity DataEC50:  54.1nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179826((R)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)p...)
Affinity DataEC50:  3nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179845(2-(4-(2-(2-chloro-4-(4-fluorophenoxy)phenoxy)ethox...)
Affinity DataEC50:  62nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179834(2-(3-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  36nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179834(2-(3-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR delta in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179834(2-(3-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  21nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179827(2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propo...)
Affinity DataEC50:  51nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179816((S)-2-(4-(3-(2-chloro-4-(4,4-dimethylcyclohexyl)ph...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR gamma in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179819(2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butox...)
Affinity DataEC50:  7.69E+3nMAssay Description:Binding affinity to human PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179844((S)-2-(4-(3-(2-chloro-4-(methylsulfonyloxy)phenoxy...)
Affinity DataEC50:  11.4nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179830((S)-2-(4-(3-(2-chloro-4-cyclohexylphenoxy)propoxy)...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR gamma in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179845(2-(4-(2-(2-chloro-4-(4-fluorophenoxy)phenoxy)ethox...)
Affinity DataEC50:  87nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179822(3-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  15nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179819(2-(4-(4-(2-chloro-4-(4-fluorophenoxy)phenoxy)butox...)
Affinity DataEC50:  66nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179835(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR delta in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179825((S)-2-((4-(3-(2,2-dimethyl-4-(3-(trifluoromethyl)p...)
Affinity DataEC50:  10nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179827(2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propo...)
Affinity DataEC50:  55nMAssay Description:Transactivation by human PPAR delta in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179818(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataEC50:  2.5nMAssay Description:Transactivation by human PPAR alpha in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50127933(CHEMBL1783044 | CHEMBL300026 | 5-(4-(3-(4-(4-fluor...)
Affinity DataEC50:  80nMAssay Description:Transactivation by human PPAR gamma in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179827(2-(4-(3-(4-(4-fluorophenoxy)-2-propylphenoxy)propo...)
Affinity DataEC50:  1.09E+3nMAssay Description:Binding affinity to human PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179828((S)-2-((4-(3-(6-chloro-2-oxo-4-(trifluoromethyl)-2...)
Affinity DataEC50: >3.00E+3nMAssay Description:Transactivation by human PPAR gamma in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179830((S)-2-(4-(3-(2-chloro-4-cyclohexylphenoxy)propoxy)...)
Affinity DataIC50: 2nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179833((S)-2-(4-(3-(2-chloro-4-(trifluoromethyl)phenoxy)p...)
Affinity DataIC50: 3nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179824((S)-2-(4-(3-(2-chloro-4-(trifluoromethoxy)phenoxy)...)
Affinity DataIC50: 3nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179818(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataIC50: 5nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179826((R)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)p...)
Affinity DataIC50: 6nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179836((S)-2-(4-(3-(2-chloro-4-(2,2,2-trifluoroethoxy)phe...)
Affinity DataIC50: 10nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179816((S)-2-(4-(3-(2-chloro-4-(4,4-dimethylcyclohexyl)ph...)
Affinity DataIC50: 22nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179829(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataIC50: 22nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179828((S)-2-((4-(3-(6-chloro-2-oxo-4-(trifluoromethyl)-2...)
Affinity DataIC50: 28nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179844((S)-2-(4-(3-(2-chloro-4-(methylsulfonyloxy)phenoxy...)
Affinity DataIC50: 30nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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