Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1466
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11558(CHEMBL381806 | (3S)-2-[(3R)-3-amino-4-(2-fluorophe...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11558(CHEMBL381806 | (3S)-2-[(3R)-3-amino-4-(2-fluorophe...)
Affinity DataIC50: 23nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50: 90nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11464(P32-98 | CHEMBL98408 | (2S,3S)-2-amino-3-methyl-1-...)
Affinity DataIC50: 140nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50: 410nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11557((2S)-1-[(3R)-3-amino-4-phenylbutanoyl]-N-({5-chlor...)
Affinity DataIC50: 1.90E+3nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 3.00E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11555((1-phenylcyclopentyl)methanamine | CHEMBL382127 | ...)
Affinity DataIC50: 3.30E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Santhera Pharmaceuticals

LigandPNGBDBM11556(2-(2-chlorophenyl)-2-(morpholin-4-yl)ethan-1-amine...)
Affinity DataIC50: 3.30E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11556(2-(2-chlorophenyl)-2-(morpholin-4-yl)ethan-1-amine...)
Affinity DataIC50: 4.60E+4nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed