Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 50017214
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179131((2E,4E)-6-(ethyl(3,5,5,8,8-pentamethyl-5,6,7,8-tet...)
Affinity DataEC50:  125nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179121((2E,4E)-3-methyl-6-((3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataEC50:  223nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179114((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  63nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179131((2E,4E)-6-(ethyl(3,5,5,8,8-pentamethyl-5,6,7,8-tet...)
Affinity DataEC50:  64nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179117((2E,4E)-6-((3,5-di-tert-butylphenyl)(methyl)amino)...)
Affinity DataEC50:  378nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179129((2E,4E)-6-((3,5-di-tert-butylphenyl)(octyl)amino)-...)
Affinity DataEC50:  35nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179125((2E,4E)-6-(ethyl(5,5,8,8-tetramethyl-5,6,7,8-tetra...)
Affinity DataEC50:  239nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179130((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  669nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179125((2E,4E)-6-(ethyl(5,5,8,8-tetramethyl-5,6,7,8-tetra...)
Affinity DataEC50:  216nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179113((2E,4E)-6-(butyl(6-tert-butyl-1,1-dimethyl-2,3-dih...)
Affinity DataEC50:  52nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179120((2E,4E)-3-methyl-6-(propyl(5,5,8,8-tetramethyl-5,6...)
Affinity DataEC50:  152nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179118((S,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  147nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179121((2E,4E)-3-methyl-6-((3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataEC50:  231nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179114((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  99nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179130((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  1.00E+3nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179115((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  100nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179120((2E,4E)-3-methyl-6-(propyl(5,5,8,8-tetramethyl-5,6...)
Affinity DataEC50:  170nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179122((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  262nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179122((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  216nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179122((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  252nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  21nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  19nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179119((2E,4E)-6-((3,5-di-tert-butylphenyl)(ethyl)amino)-...)
Affinity DataEC50:  221nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179113((2E,4E)-6-(butyl(6-tert-butyl-1,1-dimethyl-2,3-dih...)
Affinity DataEC50:  50nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179121((2E,4E)-3-methyl-6-((3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataEC50:  212nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  1.29E+3nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  22nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179115((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  123nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179117((2E,4E)-6-((3,5-di-tert-butylphenyl)(methyl)amino)...)
Affinity DataEC50:  322nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179119((2E,4E)-6-((3,5-di-tert-butylphenyl)(ethyl)amino)-...)
Affinity DataEC50:  231nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179118((S,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  161nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179115((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  98nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179118((S,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  179nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179123((2E,4E)-6-((3-methoxy-5,5,8,8-tetramethyl-5,6,7,8-...)
Affinity DataEC50:  169nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179117((2E,4E)-6-((3,5-di-tert-butylphenyl)(methyl)amino)...)
Affinity DataEC50:  95nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179131((2E,4E)-6-(ethyl(3,5,5,8,8-pentamethyl-5,6,7,8-tet...)
Affinity DataEC50:  117nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179119((2E,4E)-6-((3,5-di-tert-butylphenyl)(ethyl)amino)-...)
Affinity DataEC50:  235nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179123((2E,4E)-6-((3-methoxy-5,5,8,8-tetramethyl-5,6,7,8-...)
Affinity DataEC50:  400nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179113((2E,4E)-6-(butyl(6-tert-butyl-1,1-dimethyl-2,3-dih...)
Affinity DataEC50:  53nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179125((2E,4E)-6-(ethyl(5,5,8,8-tetramethyl-5,6,7,8-tetra...)
Affinity DataEC50:  128nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179114((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  69nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179130((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataEC50:  151nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179120((2E,4E)-3-methyl-6-(propyl(5,5,8,8-tetramethyl-5,6...)
Affinity DataEC50:  206nMAssay Description:Transactivation of RXRbeta in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179124((R,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataEC50:  1.26E+3nMAssay Description:Transactivation of RXRgamma in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataKi:  8nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataKi:  10nMAssay Description:Binding affinity to RXRgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-beta(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179116((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataKi:  12nMAssay Description:Binding affinity to RXRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179114((2E,4E)-6-((3,5-di-tert-butylphenyl)(propyl)amino)...)
Affinity DataKi:  17nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179121((2E,4E)-3-methyl-6-((3,5,5,8,8-pentamethyl-5,6,7,8...)
Affinity DataKi:  18nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179118((S,2E,4E)-3-methyl-5-(1-(5,5,8,8-tetramethyl-5,6,7...)
Affinity DataKi:  21nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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