Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50000520
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006842(CHEMBL37312 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 9.30nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006838(CHEMBL36206 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-iso...)
Affinity DataIC50: 26nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006839(CHEMBL84659 | 2-[2-(1H-Indol-3-yl)-propyl]-3-(3-is...)
Affinity DataIC50: 70nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006840(CHEMBL82690 | 2-[2-(1H-Indol-3-yl)-vinyl]-3-(3-iso...)
Affinity DataIC50: 430nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006837(CHEMBL37653 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-phenyl...)
Affinity DataIC50: 670nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006836(CHEMBL85250 | 2-[2-(5-Bromo-1H-indol-3-yl)-vinyl]-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006841(CHEMBL85393 | 2-[2-(1H-Indol-3-yl)-1-methyl-ethyl]...)
Affinity DataIC50: 9.10E+3nMAssay Description:Evaluated for inhibition of [125I]CCK-8S binding to cholecystokinin CCK-B receptor from mouse brain membranes at a concentration of 10 uM (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed