Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50003751
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475529(Clopenphendioxan)
Affinity DataKi:  0.0316nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475537(CHEMBL196817)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475534(CHEMBL198860)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475532(CHEMBL197442)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475538(CHEMBL200366)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50416853(CHEMBL43116)
Affinity DataKi:  0.0676nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475530(CHEMBL200580)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475540(CHEMBL382972)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475534(CHEMBL198860)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475533(CHEMBL199080)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475534(CHEMBL198860)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475535(CHEMBL200839)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475533(CHEMBL199080)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475538(CHEMBL200366)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475529(Clopenphendioxan)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475536(CHEMBL427552)
Affinity DataKi:  0.316nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475532(CHEMBL197442)
Affinity DataKi:  0.316nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475530(CHEMBL200580)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475533(CHEMBL199080)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475537(CHEMBL196817)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50416853(CHEMBL43116)
Affinity DataKi:  0.468nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
Affinity DataKi:  0.537nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50416853(CHEMBL43116)
Affinity DataKi:  0.537nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475535(CHEMBL200839)
Affinity DataKi:  0.562nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475532(CHEMBL197442)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475540(CHEMBL382972)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM86731(UK 33,274 | CAS_74191-85-8 | Doxazosin)
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475539(CHEMBL200136)
Affinity DataKi:  0.912nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475529(Clopenphendioxan)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475537(CHEMBL196817)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475535(CHEMBL200839)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475540(CHEMBL382972)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475536(CHEMBL427552)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475531(CHEMBL198431)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475530(CHEMBL200580)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475531(CHEMBL198431)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1D expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475536(CHEMBL427552)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475538(CHEMBL200366)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475539(CHEMBL200136)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475535(CHEMBL200839)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475531(CHEMBL198431)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1B expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475534(CHEMBL198860)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475539(CHEMBL200136)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]prazosin from cloned human ADRA1A expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475540(CHEMBL382972)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475537(CHEMBL196817)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50416853(CHEMBL43116)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475529(Clopenphendioxan)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475530(CHEMBL200580)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50475533(CHEMBL199080)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]8-hydroxy-2-(di-n-propylamino)tetralin from cloned human 5HT1A receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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