Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50017135
TargetSterol O-acyltransferase 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177892(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5,6-diphe...)
Affinity DataIC50: 940nMAssay Description:Inhibition of human ACAT1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50177891(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(6-phenyl-...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of ACAT expressed in rat liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177892(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5,6-diphe...)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human ACAT2 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177891(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(6-phenyl-...)
Affinity DataIC50: 2.07E+3nMAssay Description:Inhibition of human ACAT2 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50177892(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5,6-diphe...)
Affinity DataIC50: 2.32E+3nMAssay Description:Inhibition of ACAT expressed in rat liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177891(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(6-phenyl-...)
Affinity DataIC50: 5.34E+3nMAssay Description:Inhibition of human ACAT1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50177893(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5-phenyl-...)
Affinity DataIC50: 3.64E+4nMAssay Description:Inhibition of ACAT expressed in rat liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 2(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177893(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5-phenyl-...)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of human ACAT2 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50177893(N-(2,4-difluorophenyl)-N'-heptyl-N'-{5-[(5-phenyl-...)
Affinity DataIC50: 4.14E+5nMAssay Description:Inhibition of human ACAT1 expressed in Hi5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed